| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RPS6KA3 |
2-[4-(hydroxymethyl)anilino]-5,7-dimethyl-8-(3-methylbutyl)-7H-pteridin-6-one |
NA |
739000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
N-[(2R,3S,4S,6S)-3-methoxy-2-methyl-16-oxo-29-oxa-1,7,17-triazaoctacyclo[12.12.2.12,6.07,28.08,13.015,19.020,27.021,26]nonacosa-8,10,12,14,19,21,23,25,27-nonaen-4-yl]-N-methylbenzamide |
740000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
3-(4-amino-5-p-tolyl-7H-pyrrolo[2,3-d]pyrimidin-7-yl)propan-1-ol |
NA |
1200000|430000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KA3 |
Sunitinib |
580000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
Tozasertib |
6400000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
Dimethyl Fumarate |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
Kinase inhibitor, A1 |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA3 |
|
5600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA4 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA4 |
Pyrrolopyridine, 9 |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA4 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
2200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA4 |
Sunitinib |
2000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA5 |
2-(2-Quinolin-3-ylpyridin-4-YL)-1,5,6,7-tetrahydro-4H-pyrrolo(3,2-C)pyridin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| RPS6KA5 |
2-(2-(2-Fluorophenyl)pyridin-4-YL)-1,5,6,7-tetrahydro-4H-pyrrolo(3,2-C)pyridin-4-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| RPS6KA5 |
Pyrrolopyridine, 9 |
NA |
146000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| RPS6KA5 |
7-methoxy-3,4,5,10-tetrahydro-1H-2,5-methanoazepino[3,4-b]indole-1-carboxylic Acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| RPS6KA5 |
6-Methoxy-1,2,3,4-tetrahydro-9H-pyrido[3,4-b]indole-1-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| RPS6KA5 |
9,13-Epoxy-1H,9H-diindolo[1,2,3-gh:3',2',1'-lm]pyrrolo[3,4-j][1,7]benzodiazonin-1-one, 2,3,10,11,12,13-hexahydro-10-methoxy-9-methyl-11-(methylamino)-, (9S,10R,11R,13R)- |
890000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA5 |
Sunitinib |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| RPS6KA6 |
1H-Pyrrole-3-carboxamide, 5-((5-fluoro-1,2-dihydro-2-oxo-3H-indol-3-ylidene)methyl)-N-((2S)-2-hydroxy-3-(4-morpholinyl)propyl)-2,4-dimethyl- |
3100000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |