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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
RPS8 NB-124 sulfate NA 1493000 NA NA NA NA PubChem
RPS9 NB-124 sulfate NA 1493000 NA NA NA NA PubChem
RPSA NB-124 sulfate NA 1493000 NA NA NA NA PubChem
RRM1 [(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxy-3-methyloxolan-2-yl]methyl 2-propylpentanoate 400000 NA NA NA NA NA BindingDB
RRM1 N-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]benzenesulfonamide NA 121800 NA NA NA NA BindingDB
RRM1 N-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]-1-phenylmethanesulfonamide NA 130700 NA NA NA NA BindingDB
RRM1 benzyl N-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]carbamate NA 120300 NA NA NA NA BindingDB
RRM1 1-(7,7-dimethyl-6-oxo-2-bicyclo[2.2.1]heptanyl)-N-[(E)-(2-hydroxynaphthalen-1-yl)methylideneamino]methanesulfonamide NA 297700 NA NA NA NA BindingDB
RRM1 1-[(E)-[(E)-(4-hydroxy-3-methoxyphenyl)methylidenehydrazinylidene]methyl]naphthalen-2-ol NA 686800 NA NA NA NA BindingDB
RRM1 Hydroxyurea NA 148000|997000 NA NA NA NA BindingDB|GtoPDB|PubChem
RRM1 Ac-Tyr-Ala-Gly-Thr-Val-aIle-Ser-Asp-Leu-OH NA 395000 NA NA NA NA BindingDB
RRM1 2-{2-[2-(2-{2-[2-(2-{2-[2-Acetylamino-3-(4-hydroxy-phenyl)-propionylamino]-propionylamino}-acetylamino)-3-hydroxy-butyrylamino]-3-methyl-butyrylamino}-3-methyl-pentanoylamino)-3-carbamoyl-propionylamino]-4-carbamoyl-butyrylamino}-4-methyl-pentanoic acid NA 345000 NA NA NA NA BindingDB
RRM1 Ac-Tyr-Ala-Gly-Thr-Val-aIle-Asn-Asn-Leu-OH NA 640000 NA NA NA NA BindingDB
RRM1 Ac-Tyr-Ala-Gly-Thr-Val-aIle-Asn-Glu-Leu-OH NA 650000 NA NA NA NA BindingDB
RRM1 2-[3-Carboxy-2-(2-{3-methyl-2-[2-(3-phenyl-propionylamino)-acetylamino]-butyrylamino}-4-oxo-4-pyrrolidin-1-yl-butyrylamino)-propionylamino]-4-methyl-pentanoic acid NA 115000 NA NA NA NA BindingDB
RRM1 1-[[2-(2-{2-[(2-Benzyl-3-phenyl-propionyl)-methyl-amino]-3-methyl-butyrylamino}-3,3-dimethyl-butyrylamino)-3-carbamoyl-propionylamino]-(1-hydroxymethyl-3,3-dimethyl-butylcarbamoyl)-methyl]-cyclopentanecarboxylic acid NA NA NA 150000 NA NA BindingDB
RRM1 Val-Val-Asn-Asp-Leu NA 760000 NA NA NA NA BindingDB
RRM1 1-Aminoadenosine NA 232000|244000 NA NA NA NA BindingDB
RRM2 Hnash NA 123000 NA NA NA NA BindingDB|TTD
RRM2 Hydroxyurea NA 148000 NA NA NA NA GtoPDB|PubChem