| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| RUNX1 |
4-m-Tolyl-thiazol-2-ylamine |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| RXFP1 |
2-(cyclohexanecarbonylamino)-N-(4-methylphenyl)benzamide |
NA |
NA |
NA |
187000 |
NA |
NA |
BindingDB|TTD |
| RXRA |
2-[(E)-2-[2-cyclopropyl-4-(4-fluorophenyl)quinolin-3-yl]ethenyl]-2,3-dihydropyran-6-one |
NA |
NA |
138300 |
NA |
NA |
NA |
BindingDB |
| RXRA |
Limonene, (+/-)- |
NA |
NA |
NA |
NA |
1258930 |
NA |
PubChem |
| RXRA |
Benzene |
NA |
NA |
NA |
NA |
794328 |
NA |
PubChem |
| RXRA |
Disulfiram |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| RXRA |
Lysergide |
NA |
NA |
NA |
NA |
114057 |
NA |
PubChem |
| RXRA |
Dimethyl Sulfoxide |
NA |
NA |
NA |
NA |
19952600 |
NA |
PubChem |
| RXRA |
2-Phenylphenol |
NA |
NA |
NA |
NA |
501187|1122020 |
NA |
PubChem |
| RXRA |
2,4-Dimethylphenol |
NA |
NA |
NA |
NA |
1000000 |
NA |
PubChem |
| RXRA |
Miristalkonium chloride |
NA |
NA |
NA |
NA |
7943280 |
NA |
PubChem |
| RXRA |
Phenol |
NA |
NA |
NA |
NA |
1122020 |
NA |
PubChem |
| S100B |
5-{[(2-Mesityl-1,3-dioxo-2,3-dihydro-1h-isoindol-5-yl)carbonyl]amino}isophthalic acid |
NA |
NA |
120000 |
NA |
NA |
NA |
BindingDB |
| S1PR1 |
5-(2-Methoxypyridin-4-yl)-3-[4-(trifluoromethyl)phenyl]-1,2,4-oxadiazole |
NA |
NA |
NA |
466000 |
NA |
NA |
BindingDB |
| S1PR2 |
1-[2-(2-Hydroxyethoxy)-3-methyl-6-(trifluoromethyl)pyridin-4-yl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea |
NA |
256000 |
NA |
NA |
NA |
NA |
BindingDB |
| S1PR2 |
1-(2-Ethoxy-6-methylpyridin-4-yl)-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea |
NA |
194000 |
NA |
NA |
NA |
NA |
BindingDB |
| S1PR2 |
1-[2-(2-Hydroxyethoxy)-6-(trifluoromethyl)pyridin-4-yl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea |
NA |
348000|810000 |
NA |
NA |
NA |
NA |
BindingDB |
| S1PR2 |
1-[2-Chloro-6-(2-methoxyethoxy)pyridin-4-yl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea |
NA |
412000|3220000 |
NA |
NA |
NA |
NA |
BindingDB |
| S1PR2 |
1-[2-[2-(Dimethylamino)ethoxy]-6-(trifluoromethyl)pyridin-4-yl]-3-[[5-methyl-6-[1-methyl-3-(trifluoromethyl)pyrazol-4-yl]pyridazin-3-yl]methyl]urea |
NA |
2139000 |
NA |
NA |
NA |
NA |
BindingDB |
| S1PR2 |
1-allyl-2,5-dioxo-1,5-dihydro-2H-dipyrido[1,2-a:2',3'-d]pyrimidine-3-carbonitrile |
NA |
NA |
NA |
198300 |
NA |
NA |
BindingDB |