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      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SCN11A Dofetilide NA 300000 NA NA NA NA PubChem
SCN1A Benzocaine NA 910000 NA NA NA NA PubChem
SCN1A Caffeine NA 660000 NA NA NA NA PubChem
SCN1A Lidocaine NA 240000 NA NA NA NA PubChem
SCN1A Metoprolol NA 117000 NA NA NA NA PubChem
SCN1A Procaine NA 110000 NA NA NA NA PubChem
SCN1A (1R,3R,8S,9R,12S,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione NA 700000 NA NA NA NA PubChem
SCN1A Dofetilide NA 300000 NA NA NA NA PubChem
SCN2A 1H-Isoindole-1,3(2H)-dione, 2-(2-nitrophenyl)- 133560 NA NA NA NA NA TTD
SCN2A Benzocaine NA 910000 NA NA NA NA PubChem
SCN2A Caffeine NA 660000 NA NA NA NA PubChem
SCN2A N-(2-Carboxyphenyl)Phthalimide 337800 NA NA NA NA NA TTD
SCN2A Lidocaine NA 240000 NA NA NA NA PubChem
SCN2A Metoprolol NA 117000 NA NA NA NA PubChem
SCN2A Procaine NA 110000 NA NA NA NA PubChem
SCN2A (1R,3R,8S,9R,12S,13R,14S)-1-hydroxy-14-(2-hydroxypropan-2-yl)-13-methyl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione;(1R,3R,8S,9R,12S,13R,14R)-1-hydroxy-13-methyl-14-prop-1-en-2-yl-4,7,10-trioxapentacyclo[6.4.1.19,12.03,5.05,13]tetradecane-6,11-dione NA 700000 NA NA NA NA PubChem
SCN2A 2-(4-Methoxy-2-nitrophenyl)-1H-isoindole-1,3(2H)-dione 108070 NA NA NA NA NA TTD
SCN2A Dofetilide NA 300000 NA NA NA NA PubChem
SCN3A Benzocaine NA 910000 NA NA NA NA PubChem
SCN3A Caffeine NA 660000 NA NA NA NA PubChem