| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SELP |
3-Hydroxy-2-phenyl-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
550000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-((1H-indol-3-yl)methyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-hydroxy-8-(trifluoromethyl)quinoline-4-carboxylic acid |
NA |
325000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-hydroxy-9-(isopropylsulfonyl)-7,8,9,10-tetrahydro-1,9-phenanthroline-4-carboxylic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Hydroxy-2-(thiophen-2-ylmethyl)-7,8,9,10-tetrahydrobenzo-[h]quinoline-4-carboxylic acid |
NA |
413000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-hydroxy-8-(thien-3-yl)quinoline-4-carboxylicacid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-Benzyl-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
413000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Hydroxy-2-(thiophen-3-ylmethyl)-7,8,9,10-tetrahydrobenzo-[h]quinoline-4-carboxylic acid |
NA |
475000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Hydroxy-2-phenethyl-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chloro-benzyl)-3-hydroxy-8-phenyl-quinoline-4-carboxylic Acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(2-Chlorobenzyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]-quinoline-4-carboxylic acid |
NA |
123000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Hydroxy-2-(4-(trifluoromethoxy)benzyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
610000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-hydroxy-9-(methylsulfonyl)-7,8,9,10-tetrahydro-1,9-phenanthroline-4-carboxylic acid |
NA |
625000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
8-bromo-2-(4-chlorobenzyl)-3-hydroxyquinoline-4-carboxylic Acid |
NA |
425000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
(2S)-3-methyl-2-[[(3R,5R)-1,3,4,5-tetrahydroxycyclohexanecarbonyl]amino]pentanoic acid |
NA |
19000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
(2S)-3-hydroxy-2-[[(3R,5R)-1,3,4,5-tetrahydroxycyclohexanecarbonyl]amino]propanoic acid |
NA |
19500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-chlorobenzyl)-3-hydroxy-8-methylquinoline-4-carboxylic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
(2R)-2-[(2S,3R,4S,5S,6R)-3-benzoyloxy-2-[(2R,3R)-1,4-dimethoxy-1,4-dioxo-3-[(2S,3S,4R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxybutan-2-yl]oxy-5-hydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-3-phenylpropanoic acid |
NA |
520000|1900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
(2R)-2-[(2S,3R,4S,5S,6R)-3,5-dibenzoyloxy-2-[(2R,3R)-1,4-dimethoxy-1,4-dioxo-3-[(2S,3S,4R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxybutan-2-yl]oxy-6-(hydroxymethyl)oxan-4-yl]oxy-3-phenylpropanoic acid |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
(2R)-2-[(2S,3R,4S,5S,6R)-3-benzoyloxy-2-[(2R,3R)-1,4-dioxo-1,4-di(propan-2-yloxy)-3-[(2S,3S,4R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxybutan-2-yl]oxy-5-hydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-3-phenylpropanoic acid |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB |