| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SELP |
3-hydroxy-2-(1H-indol-3-ylmethyl)-8-isopropylquinoline-4-carboxylic acid |
NA |
415000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-((5-chloro-1H-indol-3-yl)methyl)-3-hydroxy-8-(trifluoromethyl)quinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
8-(sec-butyl)-2-(4-chlorobenzyl)-3-hydroxyquinoline-4-carboxylic Acid |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
8-Chloro-2-(4-chlorobenzyl)-3-hydroxyquinoline-4-carboxylicacid |
NA |
715000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
7-Chloro-2-(4-chlorobenzyl)-3-hydroxyquinoline-4-carboxylicacid |
NA |
900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-hydroxy-2-(1H-indol-3-ylmethyl)-8-(3-thienyl)quinoline-4-carboxylic acid |
NA |
380000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorophenylamino)-3-hydroxy-8-(trifluoromethyl)quinoline-4-carboxylic acid |
NA |
125000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
8-(4-chlorobenzyl)-7-hydroxy-2,3-dihydro-1H-9-aza-cyclopenta[a]naphthalene-6-carboxylic Acid |
NA |
580000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-Methyl-3-[2-(3,4,5-trihydroxy-phenyl)-acetylamino]-benzoic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| SELP |
(5-{2-[(3',4',5'-Trihydroxy-biphenyl-2-carbonyl)-amino]-phenyl}-thiophen-2-yl)-acetic acid |
NA |
212100 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-[1-(4-Chlorophenyl)cyclopropyl]-3-hydroxy-9-(trifluoromethyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
Rivipansel |
NA |
423000 |
NA |
NA |
NA |
NA |
GtoPDB |
| SELP |
5-Acetylamino-2-{2-[5-acetylamino-6-hydroxy-2-hydroxymethyl-4-(3,4,5-trihydroxy-tetrahydro-pyran-2-yloxy)-tetrahydro-pyran-3-yloxy]-3,5,6-trihydroxy-tetrahydro-pyran-4-yloxy}-4-hydroxy-6-(1,2,3-trihydroxy-propyl)-tetrahydro-pyran-2-carboxylic acid |
NA |
3400000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
Sodium;3,5-dihydroxy-2-[5-hydroxy-2-(hydroxymethyl)-4-(3,4,5-trihydroxy-6-methyloxan-2-yl)oxyoxan-3-yl]oxy-6-(hydroxymethyl)oxane-4-sulfonate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SELP |
2-{[1-(Methoxycarbonylmethyl-carbamoyl)-ethyl]-[2-(3,4,5-trihydroxy-6-{3-[4-(4-phenoxy-phenoxy)-phenyl]-propoxymethyl}-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
127000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-{[1-(Methoxycarbonylmethyl-carbamoyl)-ethyl]-[2-(3,4,5-trihydroxy-6-hydroxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
2-{(1-Phenethylcarbamoyl-ethyl)-[2-(3,4,5-trihydroxy-6-phenoxymethyl-tetrahydro-pyran-2-yl)-acetyl]-amino}-pentanedioic acid |
NA |
311000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
2-[2-([1-Phenethylcarbamoyl-2-(3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yl)-ethyl]-{3-[4-(4-phenoxy-phenoxy)-phenyl]-propionyl}-amino)-acetylamino]-pentanedioic acid |
NA |
283000 |
NA |
NA |
NA |
NA |
BindingDB |
| SELP |
4-[(R)-2-Hexadecanoylamino-3-(3,4,5-trihydroxy-6-methyl-tetrahydro-pyran-2-yloxy)-propionylamino]-4-methylcarbamoyl-butyric acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
sodium;[(2S,3R,4R,5R,6R)-6-[(2R,3S,4R,5S)-5-acetamido-2-(hydroxymethyl)-4-[(2S,3S,4R,5S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-3-yl]oxy-2,4,5-trihydroxyoxan-3-yl] sulfate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |