| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SELP |
Psi-697 |
NA |
125000|150000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| SELP |
3-(4-{4-[4-(2-Carboxy-vinyl)-phenyl]-5-[4-(2-dodecylcarbamoyl-vinyl)-phenyl]-1H-imidazol-2-yl}-phenyl)-isoxazole-5-carboxylic acid |
NA |
290000 |
NA |
NA |
NA |
NA |
TTD |
| SELP |
3-Hydroxy-7,8-dimethyl-2-phenylquinoline-4-carboxylic acid |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-hydroxy-2-(1H-indol-3-yl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Hydroxy-2-(5-methylthiophen-2-yl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(Benzofuran-3-ylmethyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-((5-chloro-1H-indol-3-yl)methyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-((5-bromo-1H-indol-3-yl)methyl)-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-hydroxy-2-((5-methyl-1H-indol-3-yl)methyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-hydroxy-2-((5-methoxy-1H-indol-3-yl)methyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-hydroxy-2-((2-methyl-1H-indol-3-yl)methyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
270000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Acetoxy-2-(4-chlorobenzyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
545000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-(thiophene-2-carbonyloxy)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
3-Benzoyloxy-2-[(4-chlorophenyl)methyl]-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
190000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-(cyclohexanecarbonyloxy)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-(methoxycarbonyloxy)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-(isobutoxycarbonyloxy)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-[(4-Chlorophenyl)methyl]-3-phenylmethoxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
390000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
2-(4-Chlorobenzyl)-3-hydroxy-8-isopropylquinoline-4-carboxylicacid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SELP |
6-Bromo-2-(4-chlorobenzyl)-3-hydroxyquinoline-4-carboxylicacid |
NA |
650000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |