| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTA |
1,10-Phenanthroline |
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
2,2'-Bipyridine |
NA |
100000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
Lonafarnib |
NA |
500000 |
NA |
NA |
NA |
NA |
PubChem |
| FNTA |
4-[5-(2,5-Dioxo-4-phenyl-piperazin-1-ylmethyl)-imidazol-1-ylmethyl]-benzonitrile |
NA |
950000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
11-(1-Methyl-piperidin-4-yl)-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridine |
NA |
724000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Ethylenediamine |
NA |
15500000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| FNTA |
4-(4-Methylpent-3-enyl)cyclohex-4-ene-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
2-[[4-(Dimethylamino)-6-[(2-sulfanylethylamino)methyl]-2-pyridyl]methylamino]ethanethiol |
NA |
620000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
(2S)-3-hydroxy-2-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-[(3-phenylmethoxybenzoyl)amino]butanoyl]amino]pentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Bz(4-OH)-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(2S)-3-hydroxy-2-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-[(4-phenylmethoxybenzoyl)amino]butanoyl]amino]pentanoyl]amino]propanoic acid |
NA |
166000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Bz(2-OH)-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(3-hydroxy-2-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
157000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(5-hydroxy-2-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
137000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(2-hydroxy-3-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
H-Ser-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
[(3S,4aR,6aS,12aR,12bS)-11-hydroxy-8,9-bis(hydroxymethyl)-4,4,6a,12b-tetramethyl-1,2,3,4a,5,6,12,12a-octahydrobenzo[a]xanthen-3-yl] acetate |
NA |
460000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
(E)-2-(2-{(S)-1-[(S)-1-((S)-1-Carboxy-2-hydroxy-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-2-methyl-propylcarbamoyl}-ethyl)-5,9,13-trimethyl-tetradeca-4,8,12-trienoic acid ethyl ester |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(S)-3-Hydroxy-2-{(S)-4-methyl-2-[(S)-3-methyl-2-((10E,14E)-7,11,15-trimethyl-hexadeca-6,10,14-trienoylamino)-butyrylamino]-pentanoylamino}-propionic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
4-(4,8,12-Trimethyl-tridecyl)-cyclohex-4-ene-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |