| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTB |
Thioacetic acid S-(9-methoxy-2-methyl-1,4-dioxo-1,2,3,4-tetrahydro-pyrazino[1,2-a]indol-3-yl) ester |
NA |
748000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
4-oxo-4-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]butanoic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
4-oxo-4-[[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienyl]amino]butanoic acid |
NA |
220000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Acetic acid (3S,4aR,6aS,12aR,12bS)-8,9-diformyl-11-hydroxy-4,4,6a,12b-tetramethyl-1,3,4,4a,5,6,6a,12,12a,12b-decahydro-2H-benzo[a]xanthen-3-yl ester |
NA |
560000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-[[(2S)-4-[methyl(phenylmethoxy)amino]-2-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxobutanoyl]amino]butanoyl]amino]pentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
[8-Chloro-1-(3H-imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
540000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
1-(3H-Imidazol-4-ylmethyl)-4-naphthalen-1-ylmethyl-7-phenyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine |
NA |
2968000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
[2-(2-Hydroxy-ethylsulfanyl)-phenyl]-[1-(3H-imidazol-4-ylmethyl)-7-phenyl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-methanone |
NA |
124000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
[1-(3H-Imidazol-4-ylmethyl)-9-methyl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
[7-Cyclohexyl-1-(3H-imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
186000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-4-[methyl(phenylmethoxy)amino]-4-oxobutanoyl]amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
[1-(3H-Imidazol-4-ylmethyl)-7-pyridin-2-yl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
177000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
(3,4-Dihydro-2H-quinolin-1-yl)-[1-(3H-imidazol-4-ylmethyl)-7-phenyl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-methanone |
NA |
205000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
N-[1-(3H-Imidazol-4-ylmethyl)-4-(naphthalene-1-carbonyl)-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-8-yl]-benzenesulfonamide |
NA |
249000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
[8-Amino-1-(3H-imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
1-(3H-Imidazol-4-ylmethyl)-7-phenyl-4-(1-phenyl-1H-tetrazol-5-yl)-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine |
NA |
702000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-4-[hydroxy(methyl)amino]-4-oxobutanoyl]amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]-3-hydroxypropanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[[(2S)-4-[hydroxy(methyl)amino]-2-[(2-methylpropan-2-yl)oxycarbonylamino]-4-oxobutanoyl]amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
[1-(3H-Imidazol-4-ylmethyl)-7-pyridin-3-yl-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
145000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
N'-(4-chlorophenyl)-N-cyano-1-(1H-imidazol-5-ylmethyl)-7-phenyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboximidamide |
NA |
1423000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |