| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTB |
(2R,3R)-2-Imidazol-1-ylmethyl-4-methyl-2,3-dihydro-benzo[b]thiophen-3-ol |
NA |
266000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
N-[1-(3H-Imidazol-4-ylmethyl)-4-(naphthalene-1-carbonyl)-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepin-8-yl]-acetamide |
NA |
168000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
[7-Bromo-1-(3H-imidazol-4-ylmethyl)-1,2,3,5-tetrahydro-benzo[e][1,4]diazepin-4-yl]-naphthalen-1-yl-methanone |
NA |
228000 |
NA |
NA |
NA |
NA |
BindingDB |
| FNTB |
1-(3H-Imidazol-4-ylmethyl)-4-(naphthalene-1-sulfonyl)-7-phenyl-2,3,4,5-tetrahydro-1H-benzo[e][1,4]diazepine |
NA |
426000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
(5E,9E)-6,10,14-trimethylpentadeca-5,9,13-trienoic acid |
NA |
170000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(S)-2-({(2S,3S,6S)-6-[((R)-2-Amino-3-tert-butyldisulfanyl-propionylamino)-methyl]-3-benzyloxy-tetrahydro-pyran-2-carbonyl}-amino)-4-methyl-pentanoic acid |
NA |
321000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
1,3-Isobenzofurandione, 3a,4,7,7a-tetrahydro-5-(4-methyl-3-penten-1-yl)- |
NA |
449000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
5-((E)-4,8-Dimethyl-nona-3,7-dienyl)-3a,4,7,7a-tetrahydro-isobenzofuran-1,3-dione |
NA |
190000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
1,10-Phenanthroline |
NA |
4000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
2,2'-Bipyridine |
NA |
100000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Lonafarnib |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| FNTB |
4-[5-(2,5-Dioxo-4-phenyl-piperazin-1-ylmethyl)-imidazol-1-ylmethyl]-benzonitrile |
NA |
950000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
11-(1-Methyl-piperidin-4-yl)-6,11-dihydro-5H-benzo[5,6]cyclohepta[1,2-b]pyridine |
NA |
724000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
Ethylenediamine |
NA |
15500000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FNTB |
4-(4-Methylpent-3-enyl)cyclohex-4-ene-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
2-[[4-(Dimethylamino)-6-[(2-sulfanylethylamino)methyl]-2-pyridyl]methylamino]ethanethiol |
NA |
620000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-[(3-phenylmethoxybenzoyl)amino]butanoyl]amino]pentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Bz(4-OH)-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-4-methyl-2-[[(2S)-3-methyl-2-[(4-phenylmethoxybenzoyl)amino]butanoyl]amino]pentanoyl]amino]propanoic acid |
NA |
166000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Bz(2-OH)-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |