| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(3-hydroxy-2-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
157000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(5-hydroxy-2-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
137000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2S)-3-hydroxy-2-[[(2S)-2-[[(2S)-2-[(2-hydroxy-3-phenylmethoxybenzoyl)amino]-3-methylbutanoyl]amino]-4-methylpentanoyl]amino]propanoic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
H-Ser-Val-Leu-Ser-OH |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
[(3S,4aR,6aS,12aR,12bS)-11-hydroxy-8,9-bis(hydroxymethyl)-4,4,6a,12b-tetramethyl-1,2,3,4a,5,6,12,12a-octahydrobenzo[a]xanthen-3-yl] acetate |
NA |
460000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(E)-2-(2-{(S)-1-[(S)-1-((S)-1-Carboxy-2-hydroxy-ethylcarbamoyl)-3-methyl-butylcarbamoyl]-2-methyl-propylcarbamoyl}-ethyl)-5,9,13-trimethyl-tetradeca-4,8,12-trienoic acid ethyl ester |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(S)-3-Hydroxy-2-{(S)-4-methyl-2-[(S)-3-methyl-2-((10E,14E)-7,11,15-trimethyl-hexadeca-6,10,14-trienoylamino)-butyrylamino]-pentanoylamino}-propionic acid |
NA |
360000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
4-(4,8,12-Trimethyl-tridecyl)-cyclohex-4-ene-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(4E)-4-[(2E)-3,7-dimethylocta-2,6-dienylidene]cyclohexane-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
2-[1-[(1-Oxidopyridin-1-ium-4-yl)methyl]piperidin-4-ylidene]-4-azatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene |
NA |
1832000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTB |
4-{5-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-imidazol-1-ylmethyl}-benzonitrile |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2E,5E,9E)-6,10,14-trimethylpentadeca-2,5,9,13-tetraenoic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
3-oxo-3-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propanoic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(7E,11E)-8,12,16-trimethyl-4-oxoheptadeca-7,11,15-trienoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(4E,8E)-5,9,13-trimethyltetradeca-4,8,12-trienamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(4E,8E)-N-(benzenesulfonyl)-5,9,13-trimethyltetradeca-4,8,12-trienamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
[2-Hydroxy-3-sulfanyl-1-(sulfanylmethyl)propyl] 2-(2,3-dihydro-1,4-benzodioxin-3-yl)thiazole-4-carboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
(2-Dodecenyl)succinic anhydride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Dodec-2-enylsuccinic acid |
NA |
402000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Lauric anhydride |
NA |
854000 |
NA |
NA |
NA |
NA |
TTD |