| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FOXM1 |
Troglitazone |
NA |
122400 |
NA |
NA |
NA |
NA |
PubChem |
| FPGS |
|
110000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FPGS |
4-Amino-4-deoxy-10-ethyl-10-deazapteroyl-gamma-methylene glutamic acid |
NA |
118000 |
NA |
NA |
NA |
NA |
BindingDB |
| FPGS |
2-((4-(((2,4-Diaminopteridin-6-yl)methyl)methylamino)phenyl)carbonylamino)-4-sulfobutanoic acid |
188000|198000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FPGS |
2-{4-[(2,4-Diamino-pteridin-6-ylmethyl)-methyl-amino]-benzoylamino}-3-sulfo-propionic acid |
136000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FPGS |
2-((4-(((2,4-Diaminopteridin-6-yl)methyl)methylamino)phenyl)carbonylamino)-4-phosphonobutanoic acid |
185000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FPR1 |
US10676431, Example 135 |
NA |
NA |
NA |
720000 |
NA |
NA |
BindingDB |
| FPR1 |
US10676431, Example 133 |
NA |
NA |
NA |
720000 |
NA |
NA |
BindingDB |
| FPR1 |
US10676431, Example 134 |
NA |
NA |
NA |
1500000 |
NA |
NA |
BindingDB |
| FPR1 |
US11124494, Example 73 |
NA |
NA |
NA |
330000 |
NA |
NA |
BindingDB |
| FPR1 |
1-(4-chlorophenyl)-3-[(3R)-1-[4-(2-dimethylphosphorylphenyl)-2,3-difluorophenyl]-2-oxopyrrolidin-3-yl]urea |
NA |
NA |
NA |
1500000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 2.5 |
NA |
NA |
NA |
258000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 2.3 |
NA |
NA |
NA |
223000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.6 |
NA |
NA |
NA |
523000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.7 |
NA |
NA |
NA |
166000 |
NA |
NA |
BindingDB |
| FPR2 |
2-(4,4-diethyl-2,5-dioxoimidazolidin-1-yl)-N-(4-fluorophenyl)acetamide |
NA |
NA |
NA |
2771000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.10 |
NA |
NA |
NA |
314000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.9 |
NA |
NA |
NA |
485000 |
NA |
NA |
BindingDB |
| FPR2 |
1-(4-Chlorophenyl)-3-(4-ethyl-4-methyl-2,5-dioxoimidazolidin-1-yl)urea |
NA |
NA |
NA |
157000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.12 |
NA |
NA |
NA |
860000 |
NA |
NA |
BindingDB |