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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
FSHR 5-methyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]furan-2-carboxamide NA NA NA 129000 NA NA BindingDB|TTD
FSHR N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]furan-3-carboxamide NA NA NA 494000 NA NA BindingDB|TTD
FSHR 3-methyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]furan-2-carboxamide NA NA NA 508000 NA NA BindingDB|TTD
FSHR N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]pyridine-2-carboxamide NA NA NA 185000 NA NA BindingDB|TTD
FSHR 2-methyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1,3-oxazole-4-carboxamide NA NA NA 250000 NA NA BindingDB|TTD
FSHR N-[5-[3-(2,5-dioxopyrrolidin-1-yl)propylcarbamoyl]-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide NA NA NA 184000 NA NA BindingDB|TTD
FSHR N-[5-(2-cyclopentylethylcarbamoyl)-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide NA NA NA 129000 NA NA BindingDB|TTD
FSHR N-[5-(2-aminoethylcarbamoyl)-2-[4-(2-methylphenyl)piperazin-1-yl]phenyl]furan-2-carboxamide NA NA NA 1850000 NA NA BindingDB|TTD
FSHR 2-cyclopropyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1,3-thiazole-4-carboxamide NA NA NA 184000 NA NA BindingDB|TTD
FSHR 2-cyclopropyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-(3-pyridin-4-ylpropylcarbamoyl)phenyl]-1,3-oxazole-4-carboxamide NA NA NA 153000 NA NA BindingDB|TTD
FSHR 2-cyclopropyl-N-[2-[4-(3-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1,3-oxazole-4-carboxamide NA NA NA 1440000 NA NA BindingDB|TTD
FSHR 2-cyclopropyl-N-[5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]-2-[4-[2-(trifluoromethyl)phenyl]piperazin-1-yl]phenyl]-1,3-oxazole-4-carboxamide NA NA NA 1001000 NA NA BindingDB|TTD
FSHR N-methyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]-1H-pyrrole-2-carboxamide NA NA NA 4900000 NA NA BindingDB|TTD
FTO Pyruvic Acid NA 1000000 NA NA NA NA PubChem
FTO Succinic Acid NA 370000 NA NA NA NA BindingDB|PubChem
FTO D-Glutamic Acid NA 1000000 NA NA NA NA PubChem
FTO Citric Acid NA 300000 NA NA NA NA BindingDB|PubChem
FTO Glutamic Acid NA 1000000 NA NA NA NA PubChem
FTO N-[(1R)-1-pyridin-3-ylethyl]-4-(trifluoromethoxy)benzenesulfonamide NA 285000 NA NA NA NA BindingDB
FTO (2R)-2-hydroxypentanedioic acid NA 320000|1000000 NA NA NA NA BindingDB|PubChem