| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FTO |
(2S)-2-hydroxypentanedioic acid |
NA |
320000|1000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| FTO |
Fumaric Acid |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| FTO |
(2s)-2-{[(1-Chloro-4-Hydroxyisoquinolin-3-Yl)carbonyl]amino}propanoic Acid |
NA |
110000 |
NA |
NA |
NA |
NA |
BindingDB |
| FTO |
(S)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)-3-methylbutanoic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB |
| FTO |
(R)-2-(1-chloro-4-hydroxyisoquinoline-3-carboxamido)-3-methylbutanoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| FTO |
3-[4-(2-Methylpropyl)phenyl]-1-nitrobutan-2-one |
NA |
105600 |
NA |
NA |
NA |
NA |
BindingDB |
| FTO |
Malic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FTO |
D-Lactic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FTO |
Aconitic Acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
PubChem |
| FTO |
(E)-4-oxo-4-[2-[5-(2-phenoxyphenyl)pyridine-2-carbonyl]hydrazinyl]but-2-enoic acid |
NA |
120000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2R,3S,4R,5S)-2-methylpiperidine-3,4,5-triol |
7900000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
3-Epi-fagomine |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2R,3R,4S,5S)-2-(Hydroxymethyl)piperidine-3,4,5-triol |
NA |
194000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2R,3R,4R,5S)-2-Methylpiperidine-3,4,5-triol |
1700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2S,3S,4S,5R)-2-methylpiperidine-3,4,5-triol |
1000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2R,3R,4R)-2-methyl-3,4-dihydro-2H-pyran-3,4-diol |
35000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
(2S,3R,4R,5R)-2-Hydroxymethyl-piperidine-3,4,5-triol |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
2(R), 4(R)-dihydroxypyrrolidine |
910000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
L-Fucose |
300000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| FUCA1 |
Migalastat |
34000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem |