| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FUCA1 |
ethyl 5-[(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-2-methyl-3-furoate |
NA |
200000|300000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
5-[(2R,3S,4R)-3,4-dihydroxypyrrolidin-2-yl]-N,N-diethyl-2-methyl-3-furamide |
NA |
220000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
1-Deoxymannojirimycin |
NA |
221000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
Fagomine |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUCA1 |
Sodium; Phosphoric acid mono-((3S,4S,5R)-3,4,5-trihydroxy-6-methyl-tetrahydro-thiopyran-2-yl) ester |
406000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FURIN |
N-(diaminomethylideneamino)benzamide |
376000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FURIN |
{[4-(N''-carbamimidoylhydrazinecarbonyl)phenyl]formohydrazido}methanimidamide |
173000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FURIN |
2-(1-Phenylethylidene)hydrazinecarboximidamide |
273000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FURIN |
N-[(phenylmethylidene)amino]guanidine |
500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FUT10 |
(2R,3S,4S,5R,6S)-2-[(2S,3R,4R,5R)-4,5-dihydroxy-2-(hydroxymethyl)piperidin-3-yl]oxy-6-(hydroxymethyl)oxane-3,4,5-triol |
NA |
40000000 |
NA |
NA |
NA |
NA |
BindingDB |
| FUT5 |
|
889000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| FXYD2 |
Pantoprazole |
NA |
199526 |
NA |
NA |
NA |
NA |
PubChem |
| FYN |
7-fluoro-1-methyl-9H-pyrido[3,4-b]indole |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FYN |
1-(2-Chloro-5-nitro-phenyl)-9H-beta-carboline |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FYN |
1-(5-Methyl-1H-imidazol-4-yl)-9H-beta-carboline |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| FYN |
Ac-YEEIE |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FYN |
Harmine |
NA |
250000 |
NA |
NA |
NA |
NA |
PubChem|TTD |
| FYN |
Tirabrutinib |
NA |
762000 |
NA |
NA |
NA |
NA |
PubChem |
| FYN |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
158000 |
NA |
NA |
NA |
NA |
TTD |
| FYN |
AC-Dopa-eee |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |