| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| G6PD |
5alpha-Androstan-17-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(3S,5S,8R,9S,10S,13S,14S)-3-amino-10,13-dimethyl-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-17-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
3beta-Hydroxy-16alpha,17alpha-epoxy-5alpha-pregnan-20-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(2S,3S,4S,5R,6S)-2-(2-aminoethylsulfanylmethyl)-6-methoxyoxane-3,4,5-triol |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
3-[[(2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]methylsulfonyl]propanenitrile |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(2S,3S,4S,5R,6S)-2-(3-aminopropylsulfanylmethyl)-6-methoxyoxane-3,4,5-triol |
129000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
2-amino-N-[[(2R,3S,4S,5R,6S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]methyl]ethanesulfonamide |
400000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
3-[[(2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]methylsulfanyl]propanenitrile |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
2-[2-[[(2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-methoxyoxan-2-yl]methylsulfanyl]ethyl]guanidine |
200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
N-[(3S,5S,8R,9S,10S,13S,14S)-10,13-dimethyl-17-oxo-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-3-yl]acetamide |
NA |
128000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(3S,5S,8R,9S,10S,13S,14S,17S)-10,13-dimethylspiro[1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthrene-17,2'-oxirane]-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
Bnn-20 |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
1-[(3S,5S,8S,9S,10S,13R,14S,17R)-3-hydroxy-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-17-yl]propan-2-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(3S,5S,8R,9S,10S,13S,14S,17R)-10,13-dimethylspiro[1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthrene-17,2'-oxetane]-3-ol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
1-[(3S,5S,8R,9S,10S,13S,14S,17R)-3-hydroxy-17-methoxy-10,13-dimethyl-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-17-yl]ethanone |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
3-[(3S,5S,8R,9S,10S,13S,14S)-10,13-dimethyl-17-oxo-1,2,3,4,5,6,7,8,9,11,12,14,15,16-tetradecahydrocyclopenta[a]phenanthren-3-yl]-1,1-dimethylurea |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
(3beta,5alpha)-3-Aminopregnan-20-one |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
N-[(3S,5S,8R,9S,10S,13S,14S,17S)-17-acetyl-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl]acetamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
3-[(3S,5S,8R,9S,10S,13S,14S,17S)-17-acetyl-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl]-1,1-dimethylurea |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| G6PD |
methyl N-[(3S,5S,8R,9S,10S,13S,14S,17S)-17-acetyl-10,13-dimethyl-2,3,4,5,6,7,8,9,11,12,14,15,16,17-tetradecahydro-1H-cyclopenta[a]phenanthren-3-yl]carbamate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |