| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GAA |
(2R,3R,4R,5S)-2-ethyl-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
341000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R,5S)-2-(hydroxymethyl)-2-propylpiperidine-3,4,5-triol |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2S,3S,4S)-2-(hydroxymethyl)-2-(4-hydroxyphenyl)pyrrolidine-3,4-diol |
NA |
376000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2S,3S,4S)-2-(3-fluorophenyl)-2-(hydroxymethyl)pyrrolidine-3,4-diol |
NA |
491000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(hydroxymethyl)-2-nonylpyrrolidine-3,4-diol |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(4-fluorophenyl)-2-(hydroxymethyl)pyrrolidine-3,4-diol |
NA |
714000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(hydroxymethyl)-2-(3-methoxyphenyl)pyrrolidine-3,4-diol |
NA |
776000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(hydroxymethyl)-2-(4-hydroxyphenyl)pyrrolidine-3,4-diol |
NA |
372000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2S,3S,4S)-2-(hydroxymethyl)-2-(4-methoxyphenyl)pyrrolidine-3,4-diol |
NA |
601000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R,5S)-2-(2-hydroxyethyl)-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
182000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(1R,2R,3S,9aR)-9a-(hydroxymethyl)-1,2,3,4,6,7,8,9-octahydroquinolizine-1,2,3-triol |
NA |
297000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2S,3S,4S)-2-(hydroxymethyl)-1-(4-phenylbutyl)pyrrolidine-3,4-diol |
NA |
156000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(hydroxymethyl)-1-(3-phenylpropyl)pyrrolidine-3,4-diol |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-1-heptyl-2-(hydroxymethyl)pyrrolidine-3,4-diol |
NA |
433000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-2-(hydroxymethyl)-1-(6-phenylhexyl)pyrrolidine-3,4-diol |
NA |
117000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
[(8S,9S,10R,13R,14S,17R)-17-[(E,2R,5S)-5-ethyl-6-methylhept-3-en-2-yl]-10,13-dimethyl-2,3,4,7,8,9,11,12,14,15,16,17-dodecahydro-1H-cyclopenta[a]phenanthren-3-yl] acetate |
NA |
148000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
L-ido Miglustat |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
1-Deoxynojirimycin |
NA |
192000 |
NA |
NA |
NA |
NA |
PubChem |
| GAA |
2-Benzyliminopiperidine |
3700000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GAA |
Glucobay |
NA |
817380|576200|1520000|452243|101500|320000|707900|442400|942000|817000|583600|200800 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |