| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GAA |
2-(Hydroxymethyl)-1-methyl-3,4,5-piperidinetriol |
369000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
2-Phenylamino-4,5,6,6a-tetrahydro-3aH-cyclopentaoxazole-4,5,6-triol |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
3-Anilino-5,7a-bis(hydroxymethyl)-2,4a,6,7-tetrahydrocyclopenta[b][1,4]oxazine-5,6,7-triol |
NA |
118000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
5-benzylamino-3,4-dihydro-2H-2-pyrroliumylmethanol |
4000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
6-Benzylamino-2,3,4,5-tetrahydro-2-pyridiniumylmethanol |
700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
5-Methylene-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
1-Butyl-5-methyl-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
5-Methoxy-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
1-Butyl-piperidine-3,4,5-triol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
Precose |
NA |
102000|446700|1700000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem |
| GAA |
2,5-Dideoxy-2,5-Imino-D-Glucitol |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GAA |
(3R,4s,5S)-piperidine-3,4,5-triol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
N-[5-(Adamantan-1-yl-methoxy)-pentyl]-L-altro-1-deoxynojirimycin |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GAA |
1,4-Dideoxy-1,4-imino-d-arabinitol |
115000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(1S,3R,4S,5R,6R,7S)-7-[5-(1-adamantylmethoxy)pentylamino]-3-(hydroxymethyl)-2-oxabicyclo[4.1.0]heptane-4,5-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
N-((1S,3R,4S,5R,6R,7S)-4,5-Dihydroxy-3-(hydroxymethyl)-2-oxabicyclo[4.1.0]heptan-7-yl)5-(adamant-1-yl-methoxy)pentanamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
(1S,3R,4S,5R,6R,7S)-N-butyl-4,5-dihydroxy-3-(hydroxymethyl)-2-oxabicyclo[4.1.0]heptan-7-amine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
N-((1S,3R,4S,5R,6R,7S)-4,5-Dihydroxy-3-(hydroxymethyl)-2-oxabicyclo[4.1.0]heptan-7-yl)butyramide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GAA |
6N-benzyl-2,3,4,5-tetrahydro-6-pyridiniumamine |
3700000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GAA |
(2R,3R,4R)-1-butyl-2-(hydroxymethyl)pyrrolidine-3,4-diol |
NA|258000 |
1453000|NA |
NA |
NA |
NA |
NA |
BindingDB |