Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| GAA | Miglustat | NA | 158000 | NA | NA | NA | NA | BindingDB|PubChem |
| GAA | Baicalein | NA | 500000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| GAA | (2S,3S,4S)-1-heptyl-2-(hydroxymethyl)pyrrolidine-3,4-diol | NA | 409000 | NA | NA | NA | NA | BindingDB |
| GAA | 5-Amino-1-hydroxymethyl-cyclopentane-1,2,3,4-tetraol | NA | 162000 | NA | NA | NA | NA | BindingDB |
| GAA | [(2R,3R)-4-[(2S,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)thiolan-1-ium-1-yl]-1,3-dihydroxybutan-2-yl] sulfate | NA | 3400000 | NA | NA | NA | NA | BindingDB|TTD |
| GABBR1 | 4-Amino-3-phenylbutyric acid | 177000 | NA | NA | NA | NA | NA | PubChem|TTD |
| GABBR1 | Tpmpa | NA | NA | NA | 500000 | NA | NA | BindingDB|TTD |
| GABBR1 | 4-Amino-3-phenylbutyric acid, (R)- | 177000 | NA | NA | NA | NA | NA | BindingDB |
| GABBR2 | 4-Amino-3-phenylbutyric acid | 177000 | NA | NA | NA | NA | NA | PubChem|TTD |
| GABBR2 | Tpmpa | NA | NA | NA | 500000 | NA | NA | TTD |
| GABRA1 | 2,4-Diisobutylphenol | NA | NA | NA | 251188.64 | NA | NA | BindingDB |
| GABRA1 | (4-Hydroxy-piperidin-4-yl)-phosphinic acid | 1400000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA1 | Imipenem | NA | NA | NA | NA | NA | 2000000|2400000 | PubChem |
| GABRA1 | (Piperidin-4-yl)phosphonic acid | 3300000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA1 | CID 10859491 | NA | 104000 | NA | NA | NA | NA | BindingDB |
| GABRA1 | 2,6-Dimethylphenol | NA | NA | NA | 125892.54|199526.23 | NA | NA | BindingDB |
| GABRA1 | 4-(3-(Trifluoromethyl)-3H-diazirin-3-yl)benzyl Alcohol | NA | NA|305000|465000 | NA | 700000|NA | NA | NA | BindingDB |
| GABRA1 | 2,6-Dibromophenol | NA | NA | NA | 100000000 | NA | NA | BindingDB |
| GABRA1 | 2-Amino-4-(2-methoxy-5-prop-2-enylphenyl)-6-prop-2-enylphenol | NA | NA | NA | 144300 | NA | NA | BindingDB |
| GABRA1 | (3-Aminopropyl)(n-butyl)phosphinic acid | NA | 508000 | NA | NA | NA | NA | BindingDB|PubChem |