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      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GABRA1 2,6-Diethylphenyl isothiocyanate NA NA NA 316227.77 NA NA BindingDB
GABRA1 2-Isothiocyanato-1,3-bis(propan-2-yl)benzene NA NA NA 100000000 NA NA BindingDB
GABRA1 3-(2-Chloro-4-methylphenyl)but-2-enenitrile NA NA NA 271000 NA NA BindingDB
GABRA1 Moxifloxacin NA NA NA NA NA 300000 PubChem
GABRA1 (3aS,8bS)-3,4-dimethyl-3a-phenyl-1,2-dihydropyrrolo[2,3-b]indol-8b-ol NA NA NA 110000 NA NA BindingDB
GABRA1 [2,6-Di(propan-2-yl)-4-[3-(trifluoromethyl)diazirin-3-yl]phenyl]methanol NA 460000 NA NA NA NA BindingDB
GABRA1 Delorazepam NA 555904000 NA NA NA NA PubChem
GABRA1 2-Hydroxy-3-isopropylbenzoic acid NA NA NA 100000000 NA NA BindingDB
GABRA1 Benzyl Alcohol NA NA NA 50000000 NA NA PubChem
GABRA1 Clonazepam NA 555904000 NA NA NA NA PubChem
GABRA1 Nordazepam NA 106414000 NA NA NA NA PubChem
GABRA1 Diazepam NA 123595000 NA NA NA NA PubChem
GABRA1 2,6-Dicyclopentylphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 2-Morpholin-4-yl-propionic acid 2,6-dimethoxy-phenyl ester; hydrochloride NA NA NA 198000 NA NA BindingDB
GABRA1 2,6-Di-tert-butylphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 Halazepam NA 10864300 NA NA NA NA PubChem
GABRA1 Cefazolin NA NA NA NA NA 2400000 PubChem
GABRA1 Flunitrazepam NA 263027000 NA NA NA NA PubChem
GABRA1 Isoguvacine NA NA NA 160000 NA NA BindingDB
GABRA1 Isonipecotic Acid NA NA NA 620000 NA NA BindingDB