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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
GABRA1 1H-Imidazole-5-carboxylic acid, 1-((1S)-1-phenylethyl)-, ethyl ester NA 295000 NA NA NA NA BindingDB|PubChem
GABRA1 Carumonam NA NA NA NA NA 500000 PubChem
GABRA1 Etomidate NA 577000 NA NA NA NA BindingDB|PubChem
GABRA1 2-Isopropylphenol NA NA NA 158489.32 NA NA BindingDB
GABRA1 2,6-Dimethoxyphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 2,6-Diethylphenol NA NA NA 125892.54 NA NA BindingDB
GABRA1 3,5-Di-tert-butylphenol NA NA NA 501187.23 NA NA BindingDB
GABRA1 2,4-Di-tert-butylphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 Doripenem NA NA NA NA NA 300000 PubChem
GABRA1 1,3-Diisopropylbenzene NA NA NA 100000000 NA NA BindingDB
GABRA1 3,5-Diisopropylpyrocatechol NA NA NA 199526.23 NA NA BindingDB
GABRA1 2,6-Dicyclohexylphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 2-Cyclopentylphenol NA NA NA 100000000 NA NA BindingDB
GABRA1 3-(2,4-Dichlorophenyl)butanenitrile NA NA NA 120000 NA NA BindingDB
GABRA1 N,N-dipropylbenzo[f][1,3]benzodioxole-5-carboxamide NA NA NA 102000 NA NA BindingDB
GABRA1 Piperidin-4-yl-phosphinic acid NA NA NA 270000 NA NA BindingDB
GABRA1 2,6-Diisopropylphenyl isocyanate NA NA NA 100000000 NA NA BindingDB
GABRA1 7-Aminoflunitrazepam NA 15381500 NA NA NA NA PubChem
GABRA1 Benzenethiol, 2-(1-methylethyl)- NA NA NA 100000000 NA NA BindingDB
GABRA1 Imidazoleacetic acid NA NA NA 138000|310000 NA NA BindingDB