Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| GABRA1 | Kynurenic Acid | NA | 2900000 | NA | NA | NA | NA | PubChem |
| GABRA1 | Meropenem | NA | NA | NA | NA | NA | 300000 | PubChem |
| GABRA1 | 3-Aminopropane-1-seleninic acid | NA | NA | NA | 1400000 | NA | NA | BindingDB |
| GABRA1 | Piperidine-4-Seleninic Acid | NA | NA | NA | 200000 | NA | NA | BindingDB |
| GABRA1 | Cocaine | NA | 127000 | NA | NA | NA | NA | PubChem |
| GABRA1 | Nitrazepam | NA | 100000000 | NA | NA | NA | NA | PubChem |
| GABRA1 | Benzenemethanol, 2,6-bis(1-methylethyl)- | NA | 243000 | NA | NA | NA | NA | BindingDB |
| GABRA1 | Pentobarbital | NA | 1000000 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| GABRA1 | 2,6-Diethylphenyl isocyanate | NA | NA | NA | 251188.64 | NA | NA | BindingDB |
| GABRA1 | 2-Bromo-1,3-diethylbenzene | NA | NA | NA | 125892.54 | NA | NA | BindingDB |
| GABRA1 | Amentoflavone | NA | 281838293|281838000 | NA | NA | NA | NA | BindingDB|PubChem |
| GABRA1 | 4-(2-Hydroxyethyl)-2-[3-(2-hydroxyethyl)-4-methoxyphenyl]phenol | NA | NA | NA | 105400 | NA | NA | BindingDB |
| GABRA1 | Temazepam | NA | 62517300 | NA | NA | NA | NA | PubChem |
| GABRA1 | Cefepime | NA | NA | NA | NA | NA | 2400000 | PubChem |
| GABRA1 | Ceftazidime | NA | NA | NA | NA | NA | 2400000 | PubChem |
| GABRA1 | Methyl(piperidin-4-yl)phosphinic acid | 310000 | NA | NA | NA | NA | NA | BindingDB |
| GABRA1 | Aztreonam | NA | NA | NA | NA | NA | 400000 | PubChem |
| GABRA1 | (5S)-1-methyl-5-prop-2-enyl-5-[3-[3-(trifluoromethyl)diazirin-3-yl]phenyl]-1,3-diazinane-2,4,6-trione | NA | 120000 | NA | NA | NA | NA | BindingDB|TTD |
| GABRA1 | 2,6-Dimethylthiophenol | NA | NA | NA | 100000000 | NA | NA | BindingDB |
| GABRA1 | (Z)-3-(2,4-dichlorophenyl)but-2-enenitrile | NA | NA | NA | 103000|148000|171000 | NA | NA | BindingDB |