| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FPR2 |
(2S)-3-phenyl-2-[({[4-(trifluoromethyl)phenyl]amino}carbonyl) amino]propanoic acid |
NA |
NA |
NA |
120000 |
NA |
NA |
BindingDB |
| FPR2 |
N-(4-bromophenyl)-2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)acetamide |
NA |
NA |
NA |
719000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.3 |
NA |
NA |
NA |
738000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.8 |
NA |
NA |
NA |
679000 |
NA |
NA |
BindingDB |
| FPR2 |
N-(4-bromophenyl)-2-(1,3-dioxo-1,3,3a,4,7,7a-hexahydro-2H-4,7-methanoisoindol-2-yl)acetamide |
NA |
NA |
NA |
575000 |
NA |
NA |
BindingDB |
| FPR2 |
2-(N'-(4-chlorophenyl)ureido)-3-phenylpropanoic acid |
NA |
NA |
NA |
110000 |
NA |
NA |
BindingDB |
| FPR2 |
N-(4-bromophenyl)-2-(1,3-dioxo-1,3,3a,4,7,7a-hexahydro-2H-isoindol-2-yl)acetamide |
NA |
NA |
NA |
395000 |
NA |
NA |
BindingDB |
| FPR2 |
3-Phenyl-2-[({[4-(trifluoromethoxy)phenyl]amino} carbonyl)amino]propanoic acid |
NA |
NA |
NA |
1572000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.4 |
NA |
NA |
NA |
322000 |
NA |
NA |
BindingDB |
| FPR2 |
2-({[(3,4-Dimethoxyphenyl)amino]carbonyl} amino)-3-phenylpropanoic acid |
NA |
NA |
NA |
2793000 |
NA |
NA |
BindingDB |
| FPR2 |
(2S)-2-({[(4-nitrophenyl)amino]carbonyl}amino)-3-phenylpropanoic acid |
NA |
NA |
NA |
574000 |
NA |
NA |
BindingDB |
| FPR2 |
(2S)-2-({[(4-methoxyphenyl)amino]carbonyl}amino)-3-phenylpropanoic acid |
NA |
NA |
NA |
1754000 |
NA |
NA |
BindingDB |
| FPR2 |
(2S)-2-({[(4-bromo-2-fluorophenyl)amino]carbonyl}amino)-3-methylbutanoic acid |
NA |
NA |
NA |
152000 |
NA |
NA |
BindingDB |
| FPR2 |
(2R)-2-({[(4-bromophenyl)amino]carbonyl}amino)-3-phenylpropanoic acid |
NA |
NA |
NA |
1819000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 3.5 |
NA |
NA |
NA |
645000 |
NA |
NA |
BindingDB |
| FPR2 |
(+) tert-butyl {3-[(3R)-3-(4-cyanophenyl)-7-({[4-(methylsulfinyl)phenyl] carbamoyl}amino)-1-oxo-3,4-dihydroisoquinolin-2(1H)-yl] propyl}carbamate |
NA |
NA |
NA |
103000 |
NA |
NA |
BindingDB |
| FPR2 |
US10208071, Table 2.4 |
NA |
NA |
NA |
363000 |
NA |
NA |
BindingDB |
| FSHR |
3-benzamido-4-[4-(2-methylphenyl)piperazin-1-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide |
NA |
NA |
NA |
554000 |
NA |
NA |
BindingDB|TTD |
| FSHR |
3-(cyclopropanecarbonylamino)-4-[4-(2-methylphenyl)piperazin-1-yl]-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide |
NA |
NA |
NA |
199000 |
NA |
NA |
BindingDB|TTD |
| FSHR |
N-methyl-N-[2-[4-(2-methylphenyl)piperazin-1-yl]-5-[3-(2-oxopyrrolidin-1-yl)propylcarbamoyl]phenyl]furan-2-carboxamide |
NA |
NA |
NA |
8820000 |
NA |
NA |
BindingDB|TTD |