| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTB |
tetrasodium;[2-[1-[(2E)-3,7-dimethylocta-2,6-dienyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
tetrasodium;[2-[1-[(2Z)-3,7-dimethylocta-2,6-dienyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Tetrasodium;[2-[1-(3,7-dimethylocta-2,6-dienyl)triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
Itaconic Anhydride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
tetrasodium;[2-[1-[[(2R,3R)-3-methyl-3-(4-methylpent-3-enyl)oxiran-2-yl]methyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
tetrasodium;[2-[1-[[(2R,3S)-3-methyl-3-(4-methylpent-3-enyl)oxiran-2-yl]methyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
340000 |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(2S)-2-[[[(3S,5R)-1-[(4S)-4-amino-4-carboxybutanoyl]-5-carboxypyrrolidin-3-yl]oxy-hydroxyphosphoryl]amino]pentanedioic acid |
NA |
357000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FOLH1 |
(2S)-2-[[[(3S,5R)-1-[(4S)-4-(6-aminohexanoylamino)-4-carboxybutanoyl]-5-carboxypyrrolidin-3-yl]oxy-hydroxyphosphoryl]amino]pentanedioic acid |
NA |
112000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FOLH1 |
L-Serine O-sulfate |
NA |
438000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FOLH1 |
Glutamic Acid |
NA |
428000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| FOLH1 |
(S)-3-(3-Hydroxyphenyl)-2-(3-(1-methoxy-4-methyl-1-oxopentan-2-yl)ureido)propanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-2-(3-(Carboxy(3-hydroxyphenyl)methyl)ureido)-4-methylpentanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-3-(2-Carboxy-2-(3-(1-methoxy-4-methyl-1-oxopentan-2-yl)ureido)ethyl)benzoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-2-(3-((S)-1-Methoxy-4-methyl-1-oxopentan-2-yl)ureido)-4-(methylthio)butanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-2-(3-((S)-1-Carboxy-2-(1H-indol-3-yl)ethyl)ureido)-4-methylpentanoic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-2-(4-Fluoro-3-methoxyphenyl)-2-(3-(1-methoxy-4-methyl-1-oxopentan-2-yl)ureido)acetic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
(S)-2-(3-hydroxyphenyl)-2-(3-(1-methoxy-4-methyl-1-oxopentan-2-yl)ureido)acetic acid |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| FOLH1 |
Phosphoserine |
NA |
523000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| FOLH1 |
(2S)-2-[[(1S)-1,3-dicarboxypropyl]carbamothioylamino]pentanedioic acid |
NA |
135000 |
NA |
NA |
NA |
NA |
BindingDB |
| FOS |
(1E,4Z,6E)-5-hydroxy-1,7-bis(4-hydroxy-3-methoxyphenyl)hepta-1,4,6-trien-3-one |
NA |
480000 |
NA |
NA |
NA |
NA |
PubChem |