| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| FNTA |
(4E)-4-[(2E)-3,7-dimethylocta-2,6-dienylidene]cyclohexane-1,2-dicarboxylic acid |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
2-[1-[(1-Oxidopyridin-1-ium-4-yl)methyl]piperidin-4-ylidene]-4-azatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),4,6,11,13-hexaene |
NA |
1832000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
4-{5-[4-(3-Chloro-phenyl)-piperazin-1-ylmethyl]-imidazol-1-ylmethyl}-benzonitrile |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
(2E,5E,9E)-6,10,14-trimethylpentadeca-2,5,9,13-tetraenoic acid |
NA |
130000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
3-oxo-3-[(2E,6E)-3,7,11-trimethyldodeca-2,6,10-trienoxy]propanoic acid |
NA |
160000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
(7E,11E)-8,12,16-trimethyl-4-oxoheptadeca-7,11,15-trienoic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(4E,8E)-5,9,13-trimethyltetradeca-4,8,12-trienamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(4E,8E)-N-(benzenesulfonyl)-5,9,13-trimethyltetradeca-4,8,12-trienamide |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
[2-Hydroxy-3-sulfanyl-1-(sulfanylmethyl)propyl] 2-(2,3-dihydro-1,4-benzodioxin-3-yl)thiazole-4-carboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
(2-Dodecenyl)succinic anhydride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Dodec-2-enylsuccinic acid |
NA |
402000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
Lauric anhydride |
NA |
854000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| FNTA |
tetrasodium;[2-[1-[(2E)-3,7-dimethylocta-2,6-dienyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
tetrasodium;[2-[1-[(2Z)-3,7-dimethylocta-2,6-dienyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Tetrasodium;[2-[1-(3,7-dimethylocta-2,6-dienyl)triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
Itaconic Anhydride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
tetrasodium;[2-[1-[[(2R,3R)-3-methyl-3-(4-methylpent-3-enyl)oxiran-2-yl]methyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| FNTA |
tetrasodium;[2-[1-[[(2R,3S)-3-methyl-3-(4-methylpent-3-enyl)oxiran-2-yl]methyl]triazol-4-yl]-1-phosphonatoethyl]-dioxido-oxo-lambda5-phosphane |
NA |
340000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
5-(4,8,12-Trimethyl-tridecyl)-3a,4,7,7a-tetrahydro-isobenzofuran-1,3-dione |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| FNTB |
3-[(E,E)-3,7,11-trimethyl-2,6,10-dodecatrienylamino]-3-oxo-propionic acid |
NA |
115000 |
NA |
NA |
NA |
NA |
TTD |