| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GAPDH |
N-Isopentyladenosine |
NA |
3700000 |
NA |
NA |
NA |
NA |
TTD |
| GAPDH |
N6-Benzyladenosine |
NA|2800000 |
4200000|NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GAPDH |
(2R,3S,4R)-2-(hydroxymethyl)-5-[6-[(4-hydroxy-3-methylbutyl)amino]purin-9-yl]oxolane-3,4-diol |
NA |
34003000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GAPDH |
(3R,4S,5R)-2-[6-[(4-aminophenyl)methylamino]purin-9-yl]-5-(hydroxymethyl)oxolane-3,4-diol |
NA |
3100000 |
NA |
NA |
NA |
NA |
BindingDB |
| GAPDH |
9-(2-Benzylamino-ethyl)-8-thiophen-2-yl-9H-purin-6-ylamine |
NA |
400000|500000|600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GAPDH |
2-methylpropyl N-[(2R,3R,4S,5R)-2-(6-aminopurin-9-yl)-4-hydroxy-5-(hydroxymethyl)oxolan-3-yl]carbamate |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| GART |
(2S)-2-[[4-[2-(2-amino-5,6,7,8-tetrahydropyrido[2,3-d]pyrimidin-6-yl)ethyl]benzoyl]amino]pentanedioic acid |
186000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-Methylpiperidine-3,4-diol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
8-Azabicyclo[3.2.1]octane-1,2,3,4-tetrol, (1R,2R,3R,4S,5R)- |
199000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4,5,6,7-Tetrachloro-2-(4-phenylbutyl)isoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3R,4R,5S)-2-Methylpiperidine-3,4,5-triol |
780000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3R,4R,5S,6S)-2-(hydroxymethyl)-6-propylpiperidine-3,4,5-triol |
NA |
487000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4,5,6,7-Tetrachloro-2-phenethyl-isoindole-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4,5,6,7-Tetrachloro-2-(3-phenylpropyl)isoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4-Hydroxy-2-phenylisoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4,5,6,7-Tetrachloro-2-(5-phenylpentyl)isoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-Hydroxy-2-phenylisoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-5-(Hydroxymethyl)piperidine-3,4-diol |
NA |
113000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
alpha-1-C-Propyl-DNJ |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-3,4,5-trihydroxypiperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |