| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA |
(1S,2S,3S,6R)-6-(hexylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(benzylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(octylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3S,4R,5R,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)piperidine-2-carbonitrile |
716000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-pentyl-1-deoxynojirimycin |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3S,4S)-3,4-dihydroxy-2-(hydroxymethyl)-N-octylpyrrolidine-1-carbothioamide |
NA |
121000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3R,4R)-3,4-dihydroxy-2-(hydroxymethyl)-N-octylpiperidine-1-carbothioamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3R,4R)-3,4-dihydroxy-2-(hydroxymethyl)-N-octylpyrrolidine-1-carbothioamide |
NA |
788000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,4R,5R)-4-(hydroxymethyl)-5-pyrrolidin-1-ylcyclopentane-1,2,3-triol |
123000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3S,4R)-2-[[4-[4-(hydroxymethyl)phenyl]triazol-1-yl]methyl]pyrrolidine-3,4-diol |
NA |
187000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3S,4S,5R)-1-(5-hexoxypentyl)-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
603000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3S,4S,5R)-2-(hydroxymethyl)-1-nonylpiperidine-3,4,5-triol |
NA |
136000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-(adamantan-1-yl)-4-[(2S,3R,4R,5R)-3,4-dihydroxy-2,5-bis(hydroxymethyl)pyrrolidin-1-yl]butanamide |
NA |
507000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-(adamantan-1-yl)-5-[(2S,3R,4R,5R)-3,4-dihydroxy-2,5-bis(hydroxymethyl)pyrrolidin-1-yl]pentanamide |
NA |
393000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-{2-[(3-chlorophenyl)amino]-4-methylquinolin-6-yl}-4-methylcyclohexane-1-carboxamide |
122000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
L-ido Miglustat |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-Heptyl-L-ido-1-deoxynojirimycin |
NA |
700000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
1h-Isoindole-1,3(2h)-dione, 4-nitro-2-phenyl- |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
3-Amino-N-phenylphthalimide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-phenethyl phthalimide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |