| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA |
(3S,4R,5R)-3,4,5-trihydroxy-1-(6-hydroxyhexyl)piperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5S)-1-decyl-3,4,5-trihydroxypiperidin-2-one |
NA |
295000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5S)-3,4,5-trihydroxy-1-(6-hydroxyhexyl)piperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4,5,6,7-Tetrachloro-2-(6-phenyl-hexyl)-isoindole-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
2-Anilino-6-(hydroxymethyl)-3a,4,5,6a-tetrahydrocyclopenta[d][1,3]oxazole-4,5,6-triol |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
3-Anilino-5,7a-bis(hydroxymethyl)-2,4a,6,7-tetrahydrocyclopenta[b][1,4]oxazine-5,6,7-triol |
NA |
211000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
2-anilino-4-(hydroxymethyl)-4,5,6,6a-tetrahydro-3aH-cyclopenta[d][1,3]oxazole-5,6-diol |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-Methylene-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-Methoxy-piperidine-3,4-diol |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
1-Butyl-piperidine-3,4,5-triol |
NA |
530000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
6-Hydroxymethyl-5-(3-hydroxy-pyridin-2-ylsulfanyl)-2-methoxy-tetrahydro-pyran-3,4-diol |
800000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
6-Hydroxymethyl-2-methoxy-5-(pyridin-2-ylsulfanyl)-tetrahydro-pyran-3,4-diol |
8000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-(6-Dimethylaminomethyl-3-hydroxy-pyridin-2-ylsulfanyl)-6-hydroxymethyl-2-methoxy-tetrahydro-pyran-3,4-diol |
20000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-(3-Hydroxy-6-hydroxymethyl-pyridin-2-ylsulfanyl)-6-hydroxymethyl-2-methoxy-tetrahydro-pyran-3,4-diol |
4000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
6-Hydroxymethyl-5-(3-hydroxy-6-methyl-pyridin-2-ylsulfanyl)-2-methoxy-tetrahydro-pyran-3,4-diol |
4500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-3,4,5-trihydroxy-1-nonylpiperidin-2-one |
NA |
102000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-3,4,5-trihydroxy-1-octylpiperidin-2-one |
NA |
175000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-1-butyl-3,4,5-trihydroxypiperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-1-benzyl-3,4,5-trihydroxypiperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3S,4R,5R)-3,4,5-trihydroxy-1-(2-hydroxyethyl)piperidin-2-one |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |