| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA |
(2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-triol |
380000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
1,5-Anhydro-D-Fuc-ol |
42000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(13R)-13-[(2R,3R,4R,5R)-3,4-dihydroxy-5-(hydroxymethyl)pyrrolidin-2-yl]tridecane-1,2,7,9,13-pentol |
NA |
970000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3S,4R,5S)-2-(hydroxymethyl)-1-[5-[(4-phenylphenyl)methoxy]pentyl]piperidine-3,4,5-triol |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3R,4R,5S)-2-(hydroxymethyl)-1-[5-(phenanthren-9-ylmethoxy)pentyl]piperidine-3,4,5-triol |
NA |
600000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3R,4R,5S)-2-(hydroxymethyl)-1-[5-[(1S)-1-(4-phenylphenyl)ethoxy]pentyl]piperidine-3,4,5-triol |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2S,3R,4R,5S)-1-[2,2-difluoro-5-[(4-phenylphenyl)methoxy]pentyl]-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(3aS,5R,6S,7S,7aR)-5-(hydroxymethyl)-2-(16-iodohexadecylsulfanyl)-5,6,7,7a-tetrahydro-3aH-pyrano[2,3-d][1,3]oxazole-6,7-diol |
NA |
230000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
16-[[(3aS,5R,6S,7S,7aR)-6,7-dihydroxy-5-(hydroxymethyl)-5,6,7,7a-tetrahydro-3aH-pyrano[2,3-d][1,3]oxazol-2-yl]sulfanyl]hexadecanoic acid |
NA |
420000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(decylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(3-hydroxypropylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(2-methylpropylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(2-ethylbutylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(cyclohexylmethylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(cyclohexylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(3-methylbutylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(2-phenylethylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(butylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(pentylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-6-(pentan-3-ylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |