| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA |
rel-(1R,2S,4R,5S)-6-((1-(3-(3-butoxypropoxy)propyl)-1H-1,2,3-triazol-4-yl)methylamino)cyclohexane-1,2,3,4,5-pentaol |
NA |
181000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
rel-(1R,2S,4R,5S)-6-((1-(3-(3-(3-methoxypropoxy)propoxy)propyl)-1H-1,2,3-triazol-4-yl)methylamino)cyclohexane-1,2,3,4,5-pentaol |
NA |
453000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
rel-(1R,2S,4R,5S)-6-((1-(3-(3-tert-butoxypropoxy)propyl)-1H-1,2,3-triazol-4-yl)methylamino)cyclohexane-1,2,3,4,5-pentaol |
NA |
325000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-Butoxypentyl-L-ido-1-deoxynojirimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-Pentoxypentyl-1-deoxynojirimycin |
NA |
705000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-Hexyl-L-ido-1-deoxynojirimycin |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4-Morpholin-4-ylbutane-1,3-diol |
640000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
2-Morpholinoethanol |
620000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
N-Phenylphthalimide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1R,2S,3S,4R,5S,6R)-5,6-di(nonoxy)cyclohexane-1,2,3,4-tetrol |
NA |
144000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(1S,2S,3S,6R)-4-methyl-6-(octylamino)cyclohex-4-ene-1,2,3-triol;hydrochloride |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
(2R,3S,4R,5S,6S)-5-[2-[(2S,3S,4R,5S,6R)-4,5-dihydroxy-2-(hydroxymethyl)-6-methoxyoxan-3-yl]sulfanylpyridin-3-yl]oxy-6-(hydroxymethyl)-2-methoxyoxane-3,4-diol |
5500000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GBA |
Benzylphthalimide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
4-Nitro-N-phenylphthalimide |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
2-(3-Phenyl-propyl)-isoindole-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
5-amino-2-phenyl-1H-isoindole-1,3(2H)-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
2-Benzyl-4,5,6,7-tetrachloroisoindoline-1,3-dione |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
| GBA |
Sinbaglustat |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GBA1 |
(2S,3S,4S)-1-Butyl-2-(hydroxymethyl)pyrrolidine-3,4-diol |
NA |
650000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
8-Azabicyclo[3.2.1]octane-1,2,3,4-tetrol, (1R,2R,3R,4S,5R)- |
NA|199000 |
616000|NA |
NA |
NA |
NA |
NA |
BindingDB |