| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GBA1 |
(2R,3R,4R,5S)-2-Methylpiperidine-3,4,5-triol |
780000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2S,3R,4R,5S,6S)-2-(hydroxymethyl)-6-propylpiperidine-3,4,5-triol |
NA |
487000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
Calystegine B4 |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
Ambroxol hydrochloride |
NA |
NA |
NA |
NA |
125892 |
NA |
PubChem |
| GBA1 |
(3S,4R,5R)-5-(Hydroxymethyl)piperidine-3,4-diol |
NA |
113000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
Alpha-7-Deoxyhomonojirimycin |
NA |
900000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
alpha-1-C-Propyl-DNJ |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2R,3S,4R,5R,6R)-2-butyl-6-(hydroxymethyl)piperidine-3,4,5-triol |
110000 |
100000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2S,3R,4R,5S)-2-Fluoromethyl-piperidine-3,4,5-triol |
380000|600000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
1,5-Anhydro-D-Fuc-ol |
42000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(13R)-13-[(2R,3R,4R,5R)-3,4-dihydroxy-5-(hydroxymethyl)pyrrolidin-2-yl]tridecane-1,2,7,9,13-pentol |
NA |
970000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2R,3S,4R,5S)-2-(hydroxymethyl)-1-[5-[(4-phenylphenyl)methoxy]pentyl]piperidine-3,4,5-triol |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2S,3R,4R,5S)-2-(hydroxymethyl)-1-[5-(phenanthren-9-ylmethoxy)pentyl]piperidine-3,4,5-triol |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2R,3R,4R,5S)-2-(hydroxymethyl)-1-[5-[(1S)-1-(4-phenylphenyl)ethoxy]pentyl]piperidine-3,4,5-triol |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(2S,3R,4R,5S)-1-[2,2-difluoro-5-[(4-phenylphenyl)methoxy]pentyl]-2-(hydroxymethyl)piperidine-3,4,5-triol |
NA |
500000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
methyl 16-[[(3aS,5R,6S,7S,7aR)-6,7-dihydroxy-5-(hydroxymethyl)-5,6,7,7a-tetrahydro-3aH-pyrano[2,3-d][1,3]oxazol-2-yl]sulfanyl]hexadecanoate |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
(3aS,5R,6S,7S,7aR)-5-(hydroxymethyl)-2-(16-iodohexadecylsulfanyl)-5,6,7,7a-tetrahydro-3aH-pyrano[2,3-d][1,3]oxazole-6,7-diol |
NA |
230000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
16-[[(3aS,5R,6S,7S,7aR)-6,7-dihydroxy-5-(hydroxymethyl)-5,6,7,7a-tetrahydro-3aH-pyrano[2,3-d][1,3]oxazol-2-yl]sulfanyl]hexadecanoic acid |
NA |
420000 |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
Conduritol B Epoxide |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| GBA1 |
2,5-Dideoxy-2,5-Imino-D-Mannitol |
NA |
171000 |
NA |
NA |
NA |
NA |
BindingDB |