| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GSK3B |
[2-[(5-Chloropyridin-2-yl)amino]-2-oxoethyl] 2-(4-methoxyphenyl)acetate |
NA |
NA |
NA |
107100 |
NA |
NA |
BindingDB |
| GSK3B |
Vidarabine |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
N-(5,6-diphenyl-1H-indazol-3-yl)butyramide |
NA |
1720000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
2-[4-(3-Nitro-1,2,4-triazol-1-yl)butanoylamino]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide |
NA |
NA |
NA |
105300 |
NA |
NA |
BindingDB |
| GSK3B |
Lithium Cation |
NA |
2000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| GSK3B |
2-[[5-(2,3-Dihydro-1,4-benzodioxin-3-yl)-4-methyl-1,2,4-triazol-3-yl]sulfanylmethyl]-5-(4-fluorophenyl)-1,3,4-oxadiazole |
NA |
NA |
NA |
220800 |
NA |
NA |
BindingDB |
| GSK3B |
2-[[6-Amino-2-(3-fluoroanilino)-5-nitropyrimidin-4-yl]amino]ethanol |
NA |
NA |
NA |
114000 |
NA |
NA |
BindingDB |
| GSK3B |
Ribavirin |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
2-[[6-Amino-2-[(4-methylphenyl)methylamino]-5-nitropyrimidin-4-yl]amino]ethanol |
NA |
NA |
NA |
116600 |
NA |
NA |
BindingDB |
| GSK3B |
4-Methoxypaullone |
NA |
140000|139958.73 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
4-(1H-indol-3-yl)pyrimidin-2-amine |
NA |
350000 |
NA |
NA |
NA |
NA |
BindingDB|ChEMBL |
| GSK3B |
Mefenamic Acid |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Lithium Chloride |
NA |
NA |
NA |
3000000 |
NA |
NA |
PubChem |
| GSK3B |
N-Benzyl-N'-(3-fluoro-phenyl)-5-nitro-pyrimidine-2,4,6-triamine |
NA |
NA |
NA |
108100 |
NA |
NA |
BindingDB |
| GSK3B |
2-(Thiophen-2-yl)-2,3-dihydro-1,5-benzothiazepin-4(5H)-one |
NA |
830000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
1-(4-amino-1,2,5-oxadiazol-3-yl)-5-[(2-methylpropylamino)methyl]-N-(pyridin-4-ylmethyl)triazole-4-carboxamide |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
10-Pyridin-2-yl-8-thiophen-2-yl-5,7-dihydrobenzo[d][1]benzazepine-6-thione |
NA |
349945.17 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
AR-AO-14418 |
NA |
330000 |
NA |
NA |
NA |
NA |
BindingDB |
| GSK3B |
Propyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]benzazepine-9-carboxylate |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
Pentyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]benzazepine-9-carboxylate |
NA |
600000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |