| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GSK3B |
Octyl 6-oxo-5,6,7,12-tetrahydroindolo[3,2-d][1]benzazepine-9-carboxylate |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
N-(5,6-bis(4-phenoxyphenyl)-1H-indazol-3-yl)butyramide |
NA |
10000000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
Genistein |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Chrysin |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Irsogladine Maleate |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
9-Bromo-5,6,7,12-tetrahydro-benzo[6,7]cyclohept[1,2-b]indole |
NA |
179887.09 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
9-Bromo-5,12-bis-(tert-butyloxycarbonyl)-paullone |
NA |
639734.84 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
1-[(4-methoxyphenyl)methyl]-3-[6-(2H-tetrazol-5-yl)-1,3-benzothiazol-2-yl]urea |
NA |
140000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
1-[(4-methoxyphenyl)methyl]-3-[4-(2H-tetrazol-5-yl)pyridin-2-yl]urea |
NA |
510000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
1-[(4-Methoxyphenyl)methyl]-3-(6-nitro-1,3-benzothiazol-2-yl)urea |
NA |
3640000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
1-(4-Cyanopyridin-2-yl)-3-[(4-methoxyphenyl)methyl]urea |
NA |
1430000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
Adenosine |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Tolfenamic acid |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
N-(6-Methoxy-benzothiazol-2-yl)-2-(3-methyl-3H-imidazo[4,5-b]pyridin-2-ylsulfanyl)-acetamide |
NA |
NA |
NA |
113000 |
NA |
NA |
BindingDB |
| GSK3B |
9-Chloro-7,12-dihydro-pyrido[2,3:2,3]azepino[4,5-b]-indol-6(5H)-one |
NA |
500034.53 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
12-Methyl-6-methylthio-9-nitro-7,12-dihydro-indolo-[3,2-d][1]benzazepine |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
2-[4-({[5-(pyridin-4-yl)-4H-1,2,4-triazol-3-yl]sulfanyl}methyl)phenyl]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
2-[4-({[5-(Pyridin-3-yl)-1,3,4-thiadiazol-2-yl]sulfanyl}methyl)phenyl]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
2-[4-({[5-(Pyridin-2-yl)-1,3,4-thiadiazol-2-yl]sulfanyl}methyl)phenyl]acetic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
4-{5-[(4-Iodobenzyl)sulfanyl]-1,3,4-oxadiazol-2-yl}pyridine |
NA |
198000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |