| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| GSK3B |
2-({[3-(5-Methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}sulfanyl)-5-(pyridin-4-yl)-1,3,4-oxadiazole |
NA |
250000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
Fludarabine |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
10-(3-Imidazol-1-ylpropylamino)-15-oxa-14-azatetracyclo[7.6.1.02,7.013,16]hexadeca-1(16),2,4,6,9,11,13-heptaen-8-one |
NA |
NA |
NA |
166800 |
NA |
NA |
BindingDB |
| GSK3B |
5-Cyclohexyl-4-((2-nitrobenzylidene)amino)-4H-1,2,4-triazole-3-thiol |
NA |
NA |
NA |
155000 |
NA |
NA |
BindingDB |
| GSK3B |
6-(1,9-Diazaspiro[5.5]undecan-9-Yl)-9h-Purine |
NA |
138000 |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
6-Methoxy-4-phenyl-[1]benzofuro[2,3-b]pyridin-3-ol |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
5-Methyl-2-thiophen-2-yl-2,3-dihydro-1,5-benzothiazepin-4-one |
NA |
480000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
3,6-Dimethoxy-4-phenyl-[1]benzofuro[2,3-b]pyridine |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
Propylparaben |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Butylparaben |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
Methylparaben |
NA |
NA |
NA |
300000 |
NA |
NA |
PubChem |
| GSK3B |
8-Methoxy-12-phenyl-13-phenylmethoxy-17-oxa-15-azatetracyclo[8.7.0.02,7.011,16]heptadeca-1(10),2,4,6,8,11,13,15-octaene |
1000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSK3B |
2-[[1-Cyclopentyl-5-[1-(Oxetan-3-Yl)piperidin-4-Yl]pyrazol-3-Yl]amino]pyridine-4-Carbonitrile |
NA |
682000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
(2r)-2-Methyl-1,4-Dihydropyrido[2,3-B]pyrazin-3(2h)-One |
NA |
NA |
600000|6e+05 |
NA |
NA |
NA |
BindingDB|ChEMBL |
| GSK3B |
3-({[5-(Pyridin-4-yl)-1,3,4-oxadiazol-2-yl]sulfanyl}methyl)benzoic acid |
NA |
235000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| GSK3B |
Ethyl 6-chloro-4-({4-[(2-pyrimidinylamino)sulfonyl]phenyl}amino)-3-quinolinecarboxylate |
NA |
NA |
NA |
108100 |
NA |
NA |
BindingDB |
| GSR |
3-(2-Chlorophenothiazin-10-yl)propyl-(cyclohexylmethyl)-dimethylazanium |
2000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSR |
3-(2-Chlorophenothiazin-10-yl)propyl-[(4-chlorophenyl)methyl]-dimethyl-ammonium |
2200000 |
NA |
NA |
NA |
NA |
NA |
TTD |
| GSR |
4-(Azepan-1-ylmethyl)-2,6-di-tert-butylphenol |
NA |
155000 |
NA |
NA |
NA |
NA |
TTD |
| GSR |
1-(4-(Methylsulfonyl)phenyl)-3-(piperidin-1-yl)propan-1-one |
NA |
105000 |
NA |
NA |
NA |
NA |
TTD |