| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HK2 |
(E)-3-(3,4-dichlorophenyl)-N-[(3R,4R,5S,6R)-4,5-dihydroxy-6-(hydroxymethyl)-2-methoxyoxan-3-yl]prop-2-enamide |
NA |
400000 |
NA |
NA |
NA |
NA |
TTD |
| HLCS |
[6-[(3aS,4S,6aR)-2-oxo-1,3,3a,4,6,6a-hexahydrothieno[3,4-d]imidazol-4-yl]-2-hydroxyhexyl]-[[(2R,3S,4R,5R)-5-(6-aminopurin-9-yl)-3,4-dihydroxyoxolan-2-yl]methoxy]phosphinate |
NA |
203700 |
NA |
NA |
NA |
NA |
BindingDB |
| HLCS |
Biotinol-5-amp |
754000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HMGB1 |
Glycyrrhizin |
NA |
NA |
103000|150000 |
NA |
NA |
NA |
BindingDB|PubChem |
| HMGB1 |
H-Glu-Arg-Trp-Ile-His-OH |
NA |
NA |
160000 |
NA |
NA |
NA |
BindingDB |
| HMGB1 |
5,5'-Methylenedi-2,3-cresotic acid |
NA |
NA |
900000 |
NA |
NA |
NA |
BindingDB |
| HMGB1 |
Diflunisal |
NA |
NA |
1600000 |
NA |
NA |
NA |
BindingDB|PubChem |
| HMGCR |
CID 132521485 |
NA |
387000 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
7-[(1S,2S,6S)-6-(2,2-dimethylpropanoyloxymethyl)-2-methylcyclohex-3-en-1-yl]-3,5-dihydroxyheptanoic acid |
NA |
1500000 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
Iavpgeva |
NA |
201120 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
L-Leucyl-L-prolyl-L-tyrosyl-L-proline |
NA |
484720 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
(4R,6S)-6-((E)-2-(2-cyclopropyl-6,7-difluoro-4-(3-methoxyphenylthio)quinolin-3-yl)vinyl)-4-hydroxytetrahydro-2H-pyran-2-one |
NA |
359600 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
(4R,6S)-6-((E)-2-(2-cyclopropyl-6,7-difluoro-4-(4-isopropylphenylthio)quinolin-3-yl)vinyl)-4-hydroxytetrahydro-2H-pyran-2-one |
NA |
759000 |
NA |
NA |
NA |
NA |
TTD |
| HMGCR |
Iavptgva |
NA |
152190 |
NA |
NA |
NA |
NA |
TTD |
| HOGA1 |
Dipicolinic Acid |
11000000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HOGA1 |
1,3-Phenylenediglyoxylic acid |
2960000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HOGA1 |
2-Oxoheptanedioic acid |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HOGA1 |
Chelidamic Acid |
170000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HOGA1 |
Methyl 2-[3-(2-methoxy-1-nitroso-2-oxoethyl)phenyl]-2-nitrosoacetate |
330000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HPGDS |
1-phenyl-1H-pyrazole-4-carboxylic acid |
NA |
NA|890000 |
140000|NA |
NA |
NA |
NA |
BindingDB|TTD |