| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| HPSE |
Labetalol |
NA |
NA |
1000000 |
NA |
NA |
NA |
BindingDB|PubChem |
| HPSE |
Naringin |
NA |
NA |
1000000 |
NA |
NA |
NA |
PubChem |
| HPSE |
7-chloro-N-[3-(diethylaminomethyl)-4-morpholin-4-ylphenyl]quinolin-4-amine |
NA |
NA |
239000 |
NA |
NA |
NA |
BindingDB |
| HPSE |
7-chloro-N-[4-ethoxy-3-(pyrrolidin-1-ylmethyl)phenyl]quinolin-4-amine |
NA |
NA |
169000 |
NA |
NA |
NA |
BindingDB |
| HPSE |
nonasodium;(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6R)-6-[(2R,3S,4S,5R,6R)-6-[(2R,3S,4R,5R,6S)-6-(5-aminopentoxy)-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-2-carboxylato-4-hydroxy-5-sulfonatooxyoxan-3-yl]oxy-4-hydroxy-2-(hydroxymethyl)-5-(sulfonatoamino)oxan-3-yl]oxy-3,4-dihydroxy-5-sulfonatooxyoxane-2-carboxylate |
NA |
37000000 |
NA |
NA |
NA |
NA |
BindingDB |
| HRAS |
N-[5-[[5-[(3-amino-3-iminopropyl)carbamoyl]-1-methylpyrrol-3-yl]carbamoyl]-1-methylpyrrol-3-yl]-4-formamido-1-methylpyrrole-2-carboxamide;methyl 3-[[(6aS)-2-methoxy-11-oxo-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]propanoate |
NA |
200000 |
NA |
NA |
NA |
NA |
TTD |
| HRAS |
methyl 3-[[(6aS)-2-methoxy-11-oxo-6a,7,8,9-tetrahydropyrrolo[2,1-c][1,4]benzodiazepin-3-yl]oxy]propanoate |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| HRAS |
(4S)-4-[[(2S)-2-[[(2S)-6-amino-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S)-2-[[(2S,3S)-2-[[2-[(3S,6S,11Z)-6-benzyl-3-(2-carboxyethyl)-2,5,8-trioxo-1,4,7-triazacyclotridec-11-en-1-yl]acetyl]amino]-3-methylpentanoyl]amino]-3-(4-hydroxyphenyl)propanoyl]amino]-5-carbamimidamidopentanoyl]amino]-4-methylpentanoyl]amino]-4-carboxybutanoyl]amino]-4-methylpentanoyl]amino]-4-methylpentanoyl]amino]hexanoyl]amino]propanoyl]amino]-5-[[(2S)-4-carboxy-1-[[(2S)-1-[[(2S)-1,4-diamino-1,4-dioxobutan-2-yl]amino]-1-oxopropan-2-yl]amino]-1-oxobutan-2-yl]amino]-5-oxopentanoic acid |
NA |
NA |
158000 |
NA |
NA |
NA |
BindingDB |
| HRAS |
4-[(Phenylmethoxyamino)methyl]benzene-1,2-diol |
NA |
320000 |
NA |
NA |
NA |
NA |
TTD |
| HRH1 |
Imipenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HRH1 |
(+)-(S)-N,N-dimethyl-2-(3-(1-(pyridin-2-yl)ethyl)benzo[b]thiophen-2-yl)ethanamine |
NA |
256000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| HRH1 |
1-[N'-[3-(2-amino-4-methyl-1,3-thiazol-5-yl)propyl]carbamimidoyl]-3-[(1R)-1-phenylethyl]thiourea |
109648 |
NA |
NA |
NA |
NA |
NA |
BindingDB |
| HRH1 |
Adiphenine |
NA |
112201.85|112202 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| HRH1 |
Cefazolin |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HRH1 |
Fentanyl |
NA |
147910.84|147911 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
| HRH1 |
Loratadine |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB |
| HRH1 |
Meropenem |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HRH1 |
Cefepime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HRH1 |
Ceftazidime |
NA |
NA |
NA |
NA |
NA |
300000 |
PubChem |
| HRH1 |
Aztreonam |
NA |
NA |
NA |
NA |
NA |
400000 |
PubChem |