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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HRH1 Phentolamine NA 316227.77|316228 NA NA NA NA BindingDB|PubChem|TTD
HRH1 Carumonam NA NA NA NA NA 500000 PubChem
HRH1 Doripenem NA NA NA NA NA 300000 PubChem
HRH1 Histamine 1000000|15848900000000 NA NA NA NA NA PubChem
HRH2 4-(1H-imidazol-5-yl)butan-1-amine 794328.23 NA NA NA NA NA TTD
HRH2 2,4-Pyrimidinediamine, 5-[5-iodo-4-methoxy-2-(1-methylethyl)phenoxy]- 100000000 NA NA NA NA|NA NA|NA BindingDB|TTD
HRH2 1-[N'-[3-(2-amino-1,3-thiazol-4-yl)phenyl]carbamimidoyl]-3-phenylurea 371535 NA NA NA NA NA BindingDB
HRH3 Imipenem NA NA NA NA NA 179999 PubChem
HRH3 1-[7-(3-Chlorophenoxy)heptyl]azepane 150000 NA NA NA NA NA TTD
HRH3 1-[7-(3-Chlorophenoxy)heptyl]azepane;oxalic acid 150000 NA NA NA NA NA TTD
HRH3 Cefazolin NA NA NA NA NA 300000 PubChem
HRH3 Ethyl 1-[2-(4-sulfamoylphenoxy)ethyl]piperidine-4-carboxylate NA 10000000 NA NA NA NA TTD
HRH3 Meropenem NA NA NA NA NA 300000 PubChem
HRH3 Ceftazidime NA NA NA NA NA 300000 PubChem
HRH3 Aztreonam NA NA NA NA NA 400000 PubChem
HRH3 1-Cyclohexyl-3-[4-(4-piperidin-1-ylbutoxy)phenyl]sulfonylurea NA 10000000 NA NA NA NA TTD
HRH3 Ethyl 1-[4-[4-(phenylcarbamoylsulfamoyl)phenoxy]butyl]piperidine-4-carboxylate NA 100000000 NA NA NA NA TTD
HRH3 Ethyl 1-[3-(4-sulfamoylphenoxy)propyl]piperidine-4-carboxylate NA 10000000 NA NA NA NA TTD
HRH3 Ethyl 1-[4-(4-sulfamoylphenoxy)butyl]piperidine-4-carboxylate NA 10000000 NA NA NA NA TTD
HRH3 1-Propan-2-yl-3-[4-(2-pyrrolidin-1-ylethoxy)phenyl]sulfonylurea NA 100000000 NA NA NA NA TTD