Support By : Li-lab
| GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
|---|---|---|---|---|---|---|---|---|
| HPGDS | Ethacrynic Acid | NA | 122300 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
| HPGDS | Oxfendazole | NA | 300000 | NA | NA | NA | NA | PubChem|TTD |
| HPGDS | 2-Phenyl-5-(2-phenylpyrimidin-5-yl)oxazole | NA | 125000 | NA | NA | NA | NA | BindingDB |
| HPGDS | 2-(4-Methoxybenzoyl)thiophene | NA | 105000 | NA | NA | NA | NA | BindingDB|TTD |
| HPGDS | 3-Quinolinecarbonitrile | NA | 220000 | NA | NA | NA | NA | BindingDB|TTD |
| HPN | 5-Amidinoindole | 500000 | NA | NA | NA | NA | NA | BindingDB|TTD |
| HPRT1 | {2-[(3S)-3-(2-amino-6-oxo-1,6-dihydro-9H-purin-9-yl)pyrrolidin-1-yl]-2-oxoethyl}phosphonic acid | 73000000 | NA | NA | NA | NA | NA | BindingDB |
| HPRT1 | [(3~{s},4~{r})-4-(6-Oxidanylidene-1~{h}-Purin-9-Yl)pyrrolidin-3-Yl]oxymethylphosphonic Acid | 327000 | NA | NA | NA | NA | NA | BindingDB |
| HPRT1 | 182300 | NA | NA | NA | NA | NA | BindingDB | |
| HPRT1 | 176800 | NA | NA | NA | NA | NA | BindingDB | |
| HPRT1 | 140000 | NA | NA | NA | NA | NA | BindingDB | |
| HPRT1 | 175000 | NA | NA | NA | NA | NA | BindingDB | |
| HPRT1 | 115100 | NA | NA | NA | NA | NA | BindingDB | |
| HPSE | Hesperidin | NA | NA | 1000000 | NA | NA | NA | PubChem |
| HPSE | N-[3-[(7-chloroquinolin-4-yl)amino]-5-[(4-hydroxypiperidin-1-yl)methyl]phenyl]-2-piperidin-1-ylacetamide | NA | NA | 1000000 | NA | NA | NA | BindingDB |
| HPSE | N-[3-[(7-chloroquinolin-4-yl)amino]-5-[[2-(dimethylamino)ethylamino]methyl]phenyl]-2-piperidin-1-ylacetamide | NA | NA | 639000 | NA | NA | NA | BindingDB |
| HPSE | Astemizole | NA | NA | 1000000 | NA | NA | NA | PubChem |
| HPSE | Propulsid | NA | NA | 1000000 | NA | NA | NA | PubChem |
| HPSE | 2-(3-Nitro-4-phenylsulfanylbenzoyl)benzoic acid | NA | 300000 | NA | NA | NA | NA | BindingDB|TTD |
| HPSE | Metergoline | NA | NA | 1000000 | NA | NA | NA | PubChem |