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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
HRH3 1-Cyclohexyl-3-[4-(2-pyrrolidin-1-ylethoxy)phenyl]sulfonylurea NA 10000000 NA NA NA NA TTD
HRH3 1-(2,5-Dichlorophenyl)-3-[4-(2-pyrrolidin-1-ylethoxy)phenyl]sulfonylurea NA 10000000 NA NA NA NA TTD
HRH3 1-[4-(2-Pyrrolidin-1-ylethoxy)phenyl]sulfonyl-3-[4-(trifluoromethyl)phenyl]urea NA 107000 NA NA NA NA BindingDB|TTD
HRH3 Carumonam NA NA NA NA NA 500000 PubChem
HRH3 Doripenem NA NA NA NA NA 300000 PubChem
HRH3 (4-Cyclobutylpiperazin-1-yl)-(6-cyclohexylspiro[2.5]octan-2-yl)methanone 10000000 NA NA NA NA NA TTD
HRH4 (5-Hydroxy-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 23000000|23014418 NA NA NA NA NA BindingDB
HRH4 (5,7-dimethyl-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 30900000|30974193 NA NA NA NA NA BindingDB
HRH4 (7-Amino-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 7990000|7998343 NA NA NA NA NA BindingDB
HRH4 (5-amino-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 14900000|14996848 NA NA NA NA NA BindingDB
HRH4 (7-Methyl-1H-indol-2-yl)-(4-methyl-piperazin-1-yl)-methanone 6990000|6998420 NA NA NA NA NA BindingDB
HRH4 (4,5-dichloro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 5000000|5000345 NA NA NA NA NA BindingDB
HRH4 (4-bromo-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 31900000|31988951 NA NA NA NA NA BindingDB
HRH4 1H-imidazol-5-yl(piperidin-4-yl)methanone 478000 NA NA NA NA NA BindingDB
HRH4 4-(1H-imidazol-5-yl)-1,2,3,6-tetrahydropyridine 263000 NA NA NA NA NA BindingDB
HRH4 2,4-Imidazolidinedione, 5,5-diphenyl-3-(3-(1-piperidinyl)propyl)- 489779|489778.82 NA NA NA NA NA BindingDB|TTD
HRH4 (5-methyl-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 46000000|46025657 NA NA NA NA NA BindingDB
HRH4 4-((2-Amino-6-(4-methylpiperazin-1-yl)pyrimidin-4-ylamino)methyl)benzoic acid 376600 NA NA NA NA NA BindingDB|TTD
HRH4 (5-fluoro-1H-indol-2-yl)(4-methylpiperazin-1-yl)methanone 14900000|14996848 NA NA NA NA NA BindingDB
HRH4 (5-Chloro-1H-indol-2-yl)(4-methyl-1-piperazinyl)methanone 3990000|3999447|16900000 NA NA NA NA NA BindingDB