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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACE L-leucyl-L-glutaminyl-L-proline NA 1900000 NA NA NA NA BindingDB
ACE Captopril NA NA|239883 NA 1422656|NA|1422660 NA NA BindingDB|PubChem
ACE Ac-Val-Gln-Ala-Gly-Pro-D-Ile-D-Ala-NH2 NA 2500000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-D-Ile-D-Ala-NH2 NA 850000 NA NA NA NA TTD
ACE 4-[[(2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]pyrrolidine-2-carbonyl]amino]-N-[(2R)-1-amino-1-oxopropan-2-yl]piperidine-4-carboxamide NA 10000000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-Aib-D-Ala-NH2 NA 10000000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-Gly-D-Ala-NH2 NA 2800000 NA NA NA NA TTD
ACE Ac-Val-His-Aib-Gly-Pro-D-Ile-D-Ala-NH2 NA 760000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-Gln-D-Ala-NH2 NA 1300000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-Val-D-Ala-NH2 NA 1500000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-D-Phg-D-Ala-NH2 NA 970000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-Pro-Phg-D-Ala-NH2 NA 820000 NA NA NA NA TTD
ACE (2S)-2-(3-carboxypropanoylamino)-3-methylpentanoic acid NA 1047129|1047128.55 NA NA NA NA BindingDB|TTD
ACE (2S)-1-(3-sulfanylpropyl)pyrrolidine-2-carboxylic acid NA 239883|239883.29 NA NA NA NA BindingDB|TTD
ACE (2S)-2-[(2-methyl-2-sulfanylpropanoyl)amino]butanedioic acid NA 3467369|3467368.5 NA NA NA NA BindingDB|TTD
ACE 1-(3-mercapto-propionyl)-(R)-pyrrolidine-2-carboxylic acid NA 1819701|1819700.86 NA NA NA NA BindingDB|TTD
ACE (2S)-5-oxo-1-(3-sulfanylpropyl)pyrrolidine-2-carboxylic acid NA 645654|1000000000|645654.23 NA NA NA NA BindingDB|TTD
ACE 3-(3-Sulfanylpropanoylamino)propanoic acid NA 489779|489778.82 NA NA NA NA BindingDB|TTD
ACE (2S)-2-[[(2S,3R)-2,3-dimethylpentanoyl]amino]-3-phenylpropanoic acid NA 933254|933254.3 NA NA NA NA BindingDB|TTD
ACE (2R)-1-[(2S)-2-amino-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carboxylic acid NA 181970.09 NA NA NA NA BindingDB|TTD