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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACE 5-Oxo-1-(3-sulfanylpropyl)pyrrolidine-2-carboxylic acid NA 1000000000 NA NA NA NA TTD
ACE 1-(4-Oxo-6-phenylhexanoyl)pyrrolidine-2-carboxylic acid NA 2600000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Val-Ala-NH2 NA 1500000 NA NA NA NA TTD
ACE Ac-Val-Gln-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 2500000 NA NA NA NA TTD
ACE deamino-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 2600000 NA NA NA NA TTD
ACE isovaleryl-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 165000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 850000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Ile-NHEtPh NA 325000 NA NA NA NA TTD
ACE H-Val-His-Ala-Gly-D-Pro-Ile-Ala-NH2 NA 2100000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Phg-Ala-NH2 NA 970000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-D-Phg-Ala-NH2 NA 820000 NA NA NA NA TTD
ACE H-Val-His-Ala-Gly-D-Pro-Ile-NHBn NA 260000 NA NA NA NA TTD
ACE Ac-Val-His-Val-Gly-D-Pro-Ile-Ala-NH2 NA 760000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Gly-Ala-NH2 NA 2800000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Gln-Ala-NH2 NA 1300000 NA NA NA NA TTD
ACE (2R)-N-[2-(benzylcarbamoyl)cyclopentyl]-1-[2-[[(2S)-2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]-3-methylbutanoyl]amino]acetyl]pyrrolidine-2-carboxamide NA 500000 NA NA NA NA TTD
ACE Ac-His-Ala-Gly-D-Pro-Ile-NHBn NA 280000 NA NA NA NA TTD
ACE (2R)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methylbutanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(2S,3S)-1-(3,3-diphenylpropylamino)-3-methyl-1-oxopentan-2-yl]pyrrolidine-2-carboxamide NA 365000 NA NA NA NA TTD
ACE Ac-Val-His-Ala-Gly-D-Pro-Ile-NHBn NA 115000 NA NA NA NA TTD
ACE 1-(4-carboxy-4-methylbutanoyl)-L-proline NA 260000 NA NA NA NA BindingDB|TTD