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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACE (Z)-N-[(Z)-5-(4-methoxyphenyl)-3-methylpent-2-en-4-ynoxy]-1-azabicyclo[2.2.1]heptan-3-imine NA 460000 NA NA NA NA BindingDB
ACE 2-(2-{[1-(2-{2-[2-Amino-3-(3H-imidazol-4-yl)-propionylamino]-propionylamino}-acetyl)-pyrrolidine-2-carbonyl]-amino}-3-methyl-pentanoylamino)-propionic acid NA 2000000 NA NA NA NA TTD
ACE Isoleucyl-Proline NA 128825|128000000|128824.96 NA NA NA NA BindingDB|TTD
ACE H-Pro-Val-Val-Val-Pro-Pro-OH NA 117000000 NA NA NA NA BindingDB
ACE (2S)-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]-1-[2-[[(2S)-2-[3-(1H-imidazol-5-yl)propanoylamino]propanoyl]amino]acetyl]pyrrolidine-2-carboxamide NA 10000000 NA NA NA NA TTD
ACE (2S)-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]-1-[2-[[2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]-2-methyl-propanoyl]amino]acetyl]pyrrolidine-2-carboxamide NA 10000000 NA NA NA NA TTD
ACE (2S)-N-[1-(benzylcarbamoyl)cyclopentyl]-1-[2-[[2-[[(2S)-3-(1H-imidazol-5-yl)-2-(3-methylbutanoylamino)propanoyl]amino]-2-methyl-propanoyl]amino]acetyl]pyrrolidine-2-carboxamide NA 500000 NA NA NA NA TTD
ACE Phe-Tyr NA 25100000 NA NA NA NA BindingDB
ACE His-Tyr NA 26300000 NA NA NA NA BindingDB
ACE Norathyriol NA|250200 530800|NA NA NA NA NA BindingDB|TTD
ACE Ellagic Acid NA 5000000 NA NA NA NA BindingDB|PubChem|TTD
ACE Glycyllysylproline NA 354000000 NA NA NA NA BindingDB
ACE (2S)-1-[(2S)-2-(3-phenylpropanoylamino)propanoyl]pyrrolidine-2-carboxylic acid NA 330000 NA NA NA NA TTD
ACE Novobiocin 167000 NA NA NA NA NA BindingDB|PubChem|TTD
ACE L-Alanyl-L-alanine NA 616595 NA NA NA NA BindingDB|TTD
ACE Asp-Ala NA 3801893.96 NA NA NA NA BindingDB|TTD
ACE (2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methyl-butanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[1-[[(1S)-2-amino-1-methyl-2-oxo-ethyl]carbamoyl]cyclopentyl]pyrrolidine-2-carboxamide NA 680000 NA NA NA NA TTD
ACE N-{1-[1-[1-(2-{2-[1-(1-Carbamoyl-ethylcarbamoyl)-2-methyl-butylcarbamoyl]-pyrrolidin-1-yl}-2-oxo-ethylcarbamoyl)-ethylcarbamoyl]-2-(3H-imidazol-4-yl)-ethylcarbamoyl]-2-methyl-propyl}-succinamic acid NA 1000000 NA NA NA NA TTD
ACE (2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-amino-3-methyl-butanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]pyrrolidine-2-carboxamide NA 260000 NA NA NA NA TTD
ACE (2S)-1-[2-[[(2S)-2-[[(2S)-2-[[(2S)-2-acetamido-3-methyl-butanoyl]amino]-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]pyrrolidine-2-carboxamide NA 115000 NA NA NA NA TTD