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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
ACE (2S)-1-[2-[[(2S)-2-[[(2S)-2-acetamido-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]pyrrolidine-2-carboxamide NA 280000 NA NA NA NA TTD
ACE Tyr-Ala NA 457088.19 NA NA NA NA BindingDB|TTD
ACE H-His-Ala-Gly-Pro-Ile-D-Ala-OH NA 2000000 NA NA NA NA TTD
ACE deamino-His-Ala-Gly-Pro-Ile-D-Ala-NH2 NA 2600000 NA NA NA NA TTD
ACE H-Phe-Val-Ala-Pro-OH NA 10000000 NA NA NA NA BindingDB
ACE H-Val-His-Ala-Gly-Pro-Ile-D-Ala-NH2 NA 2100000 NA NA NA NA TTD
ACE isovaleryl-His-Ala-Gly-Pro-Ile-D-Ala-NH2 NA 165000 NA NA NA NA TTD
ACE Gly-Arg NA 3235936.57 NA NA NA NA BindingDB|TTD
ACE Prolylglycine NA 16982436.52 NA NA NA NA BindingDB|TTD
ACE 2-[[(2S,3S)-2-amino-3-hydroxybutanoyl]amino]acetic acid NA 10000000 NA NA NA NA BindingDB|TTD
ACE L-Glutamyl-glycine NA 10000000 NA NA NA NA BindingDB|TTD
ACE Bucillamine NA 7244360|7244359.6 NA NA NA NA BindingDB|PubChem|TTD
ACE 3-(((1r)-1-Benzyl-2-Sulfanylethyl)Amino)-3-Oxopropanoic Acid NA 1000000000 NA NA NA NA BindingDB
ACE H-Leu-Trp-OH NA 17300000 NA NA NA NA BindingDB
ACE Met-phe NA 44600000 NA NA NA NA BindingDB
ACE H-D-Ala-phe-OH NA 190000|190546|190546.07 NA NA NA NA BindingDB|TTD
ACE Glu-Ala NA 10000000 NA NA NA NA BindingDB|TTD
ACE Gln-Gly NA 7413102.41 NA NA NA NA BindingDB|TTD
ACE H-Ile-gly-OH NA 1202264.43 NA NA NA NA BindingDB|TTD
ACE (2R)-1-[(2S,3S)-2-amino-3-methylpentanoyl]pyrrolidine-2-carboxylic acid NA 128824.96 NA NA NA NA BindingDB|TTD