Support By : Li-lab
GENE_SYMBOL | DRUG_NAME | Ki (nM) | IC50 (nM) | Kd (nM) | EC50 (nM) | Potency (nM) | AC50 (nM) | Datasource |
---|---|---|---|---|---|---|---|---|
ACE | (2S)-1-[2-[[(2S)-2-[[(2S)-2-acetamido-3-(1H-imidazol-5-yl)propanoyl]amino]propanoyl]amino]acetyl]-N-[(1S,2S)-1-(benzylcarbamoyl)-2-methyl-butyl]pyrrolidine-2-carboxamide | NA | 280000 | NA | NA | NA | NA | TTD |
ACE | Tyr-Ala | NA | 457088.19 | NA | NA | NA | NA | BindingDB|TTD |
ACE | H-His-Ala-Gly-Pro-Ile-D-Ala-OH | NA | 2000000 | NA | NA | NA | NA | TTD |
ACE | deamino-His-Ala-Gly-Pro-Ile-D-Ala-NH2 | NA | 2600000 | NA | NA | NA | NA | TTD |
ACE | H-Phe-Val-Ala-Pro-OH | NA | 10000000 | NA | NA | NA | NA | BindingDB |
ACE | H-Val-His-Ala-Gly-Pro-Ile-D-Ala-NH2 | NA | 2100000 | NA | NA | NA | NA | TTD |
ACE | isovaleryl-His-Ala-Gly-Pro-Ile-D-Ala-NH2 | NA | 165000 | NA | NA | NA | NA | TTD |
ACE | Gly-Arg | NA | 3235936.57 | NA | NA | NA | NA | BindingDB|TTD |
ACE | Prolylglycine | NA | 16982436.52 | NA | NA | NA | NA | BindingDB|TTD |
ACE | 2-[[(2S,3S)-2-amino-3-hydroxybutanoyl]amino]acetic acid | NA | 10000000 | NA | NA | NA | NA | BindingDB|TTD |
ACE | L-Glutamyl-glycine | NA | 10000000 | NA | NA | NA | NA | BindingDB|TTD |
ACE | Bucillamine | NA | 7244360|7244359.6 | NA | NA | NA | NA | BindingDB|PubChem|TTD |
ACE | 3-(((1r)-1-Benzyl-2-Sulfanylethyl)Amino)-3-Oxopropanoic Acid | NA | 1000000000 | NA | NA | NA | NA | BindingDB |
ACE | H-Leu-Trp-OH | NA | 17300000 | NA | NA | NA | NA | BindingDB |
ACE | Met-phe | NA | 44600000 | NA | NA | NA | NA | BindingDB |
ACE | H-D-Ala-phe-OH | NA | 190000|190546|190546.07 | NA | NA | NA | NA | BindingDB|TTD |
ACE | Glu-Ala | NA | 10000000 | NA | NA | NA | NA | BindingDB|TTD |
ACE | Gln-Gly | NA | 7413102.41 | NA | NA | NA | NA | BindingDB|TTD |
ACE | H-Ile-gly-OH | NA | 1202264.43 | NA | NA | NA | NA | BindingDB|TTD |
ACE | (2R)-1-[(2S,3S)-2-amino-3-methylpentanoyl]pyrrolidine-2-carboxylic acid | NA | 128824.96 | NA | NA | NA | NA | BindingDB|TTD |