GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SELP |
6-deoxy-Hex(?1-3)[Hex3S(?1-4)]Hex |
NA |
300000 |
NA |
NA |
NA |
NA |
BindingDB |
SELP |
2-[3-[2-[(2R,3S,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxyphenyl]phenyl]acetic acid |
NA |
500000 |
NA |
NA |
NA |
NA |
TTD |
SELPLG |
Oxycinchophen |
NA |
6000000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SELPLG |
2-Benzyl-3-hydroxy-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
413000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
Psi-697 |
NA |
150000 |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SELPLG |
3-Hydroxy-2-(4-hydroxyphenyl)-7,8-dimethylquinoline-4-carboxylicacid |
NA |
3500000 |
NA |
NA |
NA |
NA |
TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxyquinoline-4-carboxylic acid |
NA |
4000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
6-Bromo-2-(4-chlorophenyl)-3-hydroxyquinoline-4-carboxylicacid |
NA |
1000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
8-(4-Carboxyphenyl)-2-(4-chlorophenyl)-3-hydroxyquinoline-4-carboxylic acid |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3,6-dihydroxyquinoline-4-carboxylic acid |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
6-Amino-2-(4-chlorophenyl)-3-hydroxyquinoline-4-carboxylicacid |
NA |
3000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-7,8-dimethylquinoline-4-carboxylicacid |
NA |
450000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Bromophenyl)-3-hydroxy-7,8-dimethylquinoline-4-carboxylicacid |
NA |
400000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-8-trifluoromethylquinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-8-methylquinoline-4-carboxylicacid |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-8-isopropylquinoline-4-carboxylicacid |
NA |
225000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-7-isopropylquinoline-4-carboxylicacid |
NA |
1500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-8-phenylquinoline-4-carboxylic acid |
NA |
200000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-7-phenylquinoline-4-carboxylicacid |
NA |
2000000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-Chlorophenyl)-3-hydroxy-6-phenylquinoline-4-carboxylic acid |
NA |
375000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |