GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SELPLG |
3-Hydroxy-2-(4-isopropylphenyl)-7,8-dimethylquinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
2-(4-(Diethylamino)phenyl)-3-hydroxy-7,8-dimethylquinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
3-Hydroxy-2-(1-phenylcyclopropyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
250000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
5-Acetylamino-2-{2-[5-acetylamino-6-hydroxy-2-hydroxymethyl-4-(3,4,5-trihydroxy-tetrahydro-pyran-2-yloxy)-tetrahydro-pyran-3-yloxy]-3,5,6-trihydroxy-tetrahydro-pyran-4-yloxy}-4-hydroxy-6-(1,2,3-trihydroxy-propyl)-tetrahydro-pyran-2-carboxylic acid |
NA |
15000000 |
NA |
NA |
NA |
NA |
BindingDB |
SELPLG |
(4R,5S)-2-[(3S,4S,5S)-2-[(2S,3S)-5-acetamido-6-hydroxy-2-(hydroxymethyl)-4-[(2S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-3-yl]oxy-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-5-[[6-[2-[[(1S)-1,3-dicarboxypropyl]amino]-2-oxoethyl]-3,4,5-trihydroxyoxan-2-yl]methylcarbamoylamino]-4-hydroxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]oxane-2-carboxylate |
NA |
250000000 |
NA |
NA |
NA |
NA |
BindingDB |
SELPLG |
2-[2-(3,4,5-Trihydroxy-6-{[2-(1-phenyl-ethylcarbamoyl)-benzoylamino]-methyl}-tetrahydro-pyran-2-yl)-acetylamino]-pentanedioic acid |
NA |
2500000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
3-Hydroxy-2-(1-phenylethyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid |
NA |
175000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SELPLG |
|
NA |
3500000 |
NA |
NA |
NA |
NA |
BindingDB |
SELPLG |
Sialyl Lewis X Antigen |
NA |
15000000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(3,4-dihydroxybenzenesulfonamide) |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,4-dihydroxybenzenesulfonamide) |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N-(3,4-dihydroxyphenylsulfonyl)-N-hexyl-3,4-dihydroxybenzenesulfonamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N-cyclohexyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxybenzenesulfonamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-4-hydroxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-2,5-dihydroxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethylbenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,5-difluoro-4-hydroxybenzenesulfonamide) |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxy-N-propylbenzenesulfonamide |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N-benzyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxybenzenesulfonamide |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,4-dimethoxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |