Navigator

      Support By : Li-lab

Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SELPLG 3-Hydroxy-2-(4-isopropylphenyl)-7,8-dimethylquinoline-4-carboxylic acid NA 250000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-(Diethylamino)phenyl)-3-hydroxy-7,8-dimethylquinoline-4-carboxylic acid NA 250000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-2-(1-phenylcyclopropyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid NA 250000 NA NA NA NA BindingDB|TTD
SELPLG 5-Acetylamino-2-{2-[5-acetylamino-6-hydroxy-2-hydroxymethyl-4-(3,4,5-trihydroxy-tetrahydro-pyran-2-yloxy)-tetrahydro-pyran-3-yloxy]-3,5,6-trihydroxy-tetrahydro-pyran-4-yloxy}-4-hydroxy-6-(1,2,3-trihydroxy-propyl)-tetrahydro-pyran-2-carboxylic acid NA 15000000 NA NA NA NA BindingDB
SELPLG (4R,5S)-2-[(3S,4S,5S)-2-[(2S,3S)-5-acetamido-6-hydroxy-2-(hydroxymethyl)-4-[(2S,6S)-3,4,5-trihydroxy-6-methyloxan-2-yl]oxyoxan-3-yl]oxy-3,5-dihydroxy-6-(hydroxymethyl)oxan-4-yl]oxy-5-[[6-[2-[[(1S)-1,3-dicarboxypropyl]amino]-2-oxoethyl]-3,4,5-trihydroxyoxan-2-yl]methylcarbamoylamino]-4-hydroxy-6-[(1R,2R)-1,2,3-trihydroxypropyl]oxane-2-carboxylate NA 250000000 NA NA NA NA BindingDB
SELPLG 2-[2-(3,4,5-Trihydroxy-6-{[2-(1-phenyl-ethylcarbamoyl)-benzoylamino]-methyl}-tetrahydro-pyran-2-yl)-acetylamino]-pentanedioic acid NA 2500000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-2-(1-phenylethyl)-7,8,9,10-tetrahydrobenzo[h]quinoline-4-carboxylic acid NA 175000 NA NA NA NA BindingDB|TTD
SELPLG NA 3500000 NA NA NA NA BindingDB
SELPLG Sialyl Lewis X Antigen NA 15000000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(3,4-dihydroxybenzenesulfonamide) NA 3000000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,4-dihydroxybenzenesulfonamide) NA 1000000 NA NA NA NA TTD
SERPINC1 N-(3,4-dihydroxyphenylsulfonyl)-N-hexyl-3,4-dihydroxybenzenesulfonamide NA 300000 NA NA NA NA TTD
SERPINC1 N-cyclohexyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxybenzenesulfonamide NA 300000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-4-hydroxybenzenesulfonamide) NA 300000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-2,5-dihydroxybenzenesulfonamide) NA 300000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethylbenzenesulfonamide) NA 300000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,5-difluoro-4-hydroxybenzenesulfonamide) NA 3000000 NA NA NA NA TTD
SERPINC1 N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxy-N-propylbenzenesulfonamide NA 1000000 NA NA NA NA TTD
SERPINC1 N-benzyl-N-(3,4-dihydroxyphenylsulfonyl)-3,4-dihydroxybenzenesulfonamide NA 300000 NA NA NA NA TTD
SERPINC1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,4-dimethoxybenzenesulfonamide) NA 300000 NA NA NA NA TTD