| GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
| SERPINC1 |
N,N''-(butane-1,4-diyl)bis(3,4-dihydroxybenzenesulfonamide) |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINC1 |
N,N''-(hexane-1,6-diyl)bis(3,4-dihydroxybenzenesulfonamide) |
NA |
3000000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINC1 |
N,N''-bis(3,4-dihydroxybenzenesulfonyl)piperazine |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINC1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3-hydroxybenzenesulfonamide) |
NA |
1000000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINE1 |
N,N''-1,3-Propanediylbis(3,4,5-trihydroxybenzamide)Hydrate |
NA |
269000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
N,N''-1,2-Ethanediylbis(3,4,5-trihydroxybenzamide)Hydrate |
NA |
900000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
euglobal IIC |
NA |
700000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
US9120744, Cde-072 |
NA |
104000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
US9120744, Cde-012 |
NA |
196000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
2-[N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-4-[[2-(trifluoromethoxy)phenyl]sulfonylamino]anilino]-2-oxoacetic acid |
NA |
114000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
US9120744, Cde-011 |
NA |
338000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
Boc-3-nitro-L-tyrosine |
NA |
386000 |
NA |
NA |
NA |
NA |
BindingDB |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(3,4-dihydroxybenzenesulfonamide) |
NA |
450000|518000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
(7R,8aR,9S,10aR)-1,3-dihydroxy-10a-methyl-9-(2-methylpropyl)-7-propan-2-yl-7,8,8a,9-tetrahydroxanthene-2,4-dicarbaldehyde |
NA |
138000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
(1'S,2R,4R,5'R)-5,7-dihydroxy-6',6'-dimethyl-4-(2-methylpropyl)spiro[3,4-dihydrochromene-2,2'-bicyclo[3.1.1]heptane]-6,8-dicarbaldehyde |
NA |
152000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-4-hydroxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-2,5-dihydroxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(N-ethylbenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,5-difluoro-4-hydroxybenzenesulfonamide) |
NA |
128000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
| SERPINE1 |
N,N''-(ethane-1,2-diyl)bis(N-ethyl-3,4-dimethoxybenzenesulfonamide) |
NA |
300000 |
NA |
NA |
NA |
NA |
TTD |