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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SERPINE1 N,N''-(butane-1,4-diyl)bis(3,4-dihydroxybenzenesulfonamide) NA 3000000 NA NA NA NA TTD
SERPINE1 N,N''-(hexane-1,6-diyl)bis(3,4-dihydroxybenzenesulfonamide) NA 1384000 NA NA NA NA BindingDB|TTD
SERPINE1 N,N''-bis(3,4-dihydroxybenzenesulfonyl)piperazine NA 300000 NA NA NA NA TTD
SERPINE1 N,N''-(ethane-1,2-diyl)bis(N-ethyl-3-hydroxybenzenesulfonamide) NA 343000 NA NA NA NA BindingDB|TTD
SERPINE1 US9120744, Cde-060 NA 236000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-035 NA 146000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-061 NA 332000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-033 NA 246000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-064 NA 2204000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-057 NA 195000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-065 NA 423000 NA NA NA NA BindingDB
SERPINE1 US9120744, Cde-069 NA 562000 NA NA NA NA BindingDB
SERPINE1 (Z)-3-((Z)-Benzylidene)-6-((5-((2-(dimethylamino)ethyl)thio)thiophen-2-yl)methylene)piperazine-2,5-dione NA 106000 NA NA NA NA BindingDB
SETD7 DC_05 NA 150000 NA NA NA NA TTD
SETD7 4-methyl-3-nitro-N-(3-nitrophenyl)benzamide NA 189700 NA NA NA NA TTD
SETD7 Carm1-IN-1 NA 667000 NA NA NA NA TTD
SETD7 Kaempferol NA 200000 NA NA NA NA PubChem
SETD7 (3E,5E)-3,5-bis[(3-bromo-4-hydroxyphenyl)methylidene]-1-[(3-chlorophenyl)methyl]piperidin-4-one NA 174000 NA NA NA NA TTD
SETD7 (3E,5E)-3,5-bis[(3-bromo-4-hydroxyphenyl)methylidene]-1-phenacylpiperidin-4-one NA 149000 NA NA NA NA TTD
SETD7 (3E,5E)-3,5-bis[(3-bromo-4-hydroxyphenyl)methylidene]-1-[(2-methylphenyl)methyl]piperidin-4-one NA 667000 NA NA NA NA TTD