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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-6-(trifluoromethoxy)quinoline-4-carboxylic acid NA 625000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-phenylquinoline-4-carboxylic acid NA 1500000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-p-tolylquinoline-4-carboxylic acid NA 1000000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-(4-morpholinophenyl)quinoline-4-carboxylic acid NA 1000000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-(3-(trifluoromethoxy)phenyl)quinoline-4-carboxylic acid NA 200000 NA NA NA NA BindingDB|TTD
SELPLG 2-(3-Chlorophenyl)-3-hydroxy-7,8-dimethylquinoline-4-carboxylicacid NA 400000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-8-(4-hydroxymethylphenyl)-quinoline-4-carboxylic acid NA 2000000 NA NA NA NA BindingDB|TTD
SELPLG 6-Bromo-2-(4-chlorophenyl)-3-hydroxy-8-methylquinoline-4-carboxylic acid NA 125000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-(4-(trifluoromethyl)phenyl)quinoline-4-carboxylic acid NA 300000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-7,8-dimethyl-2-(4-(trifluoromethoxy)phenyl) quinoline-4-carboxylic acid NA 240000 NA NA NA NA BindingDB|TTD
SELPLG 3-Hydroxy-2-(4-methoxyphenyl)-7,8-dimethylquinoline-4-carboxylic acid NA 1000000 NA NA NA NA BindingDB|TTD
SELPLG 8-Chloro-2-(4-chlorophenyl)-3-hydroxyquinoline-4-carboxylicacid NA 600000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-8-(trifluoromethoxy)quinoline-4-carboxylic acid NA 550000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-6-(trifluoromethyl)quinoline-4-carboxylic acid NA 1600000 NA NA NA NA BindingDB|TTD
SELPLG 8-Bromo-2-(4-chlorophenyl)-3-hydroxyquinoline-4-carboxylicacid NA 625000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-8-(dimethylaminophenyl)-3-hydroxyquinoline-4-carboxylic acid NA 300000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-8-ethyl-3-hydroxyquinoline-4-carboxylicacid NA 525000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-8-(thien-3-yl)quinoline-4-carboxylicacid NA 175000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-6,8-dimethylquinoline-4-carboxylicacid NA 500000 NA NA NA NA BindingDB|TTD
SELPLG 2-(4-Chlorophenyl)-3-hydroxy-8-methyl-6-(trifluoromethoxy)-quinoline-4-carboxylic acid NA 225000 NA NA NA NA BindingDB|TTD