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Drugs And Genes
Negative Drug Target Genes
GENE_SYMBOL DRUG_NAME Ki (nM) IC50 (nM) Kd (nM) EC50 (nM) Potency (nM) AC50 (nM) Datasource
SLC15A1 Arg-Arg NA 7310000 NA NA NA NA BindingDB|TTD
SLC15A1 Pro-Tyr 730000 NA NA NA NA NA TTD
SLC15A1 Ala-Ser 140000 NA NA NA NA NA BindingDB|TTD
SLC15A1 Glycyl-L-alanine NA NA|1820000 NA 520000|NA NA NA BindingDB|TTD
SLC15A1 [(3S,7R,8aS)-7-hydroxy-1,4-dioxo-2,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-3-yl]methyl (2S)-2-amino-3-methylbutanoate NA 2900000 NA NA NA NA BindingDB|TTD
SLC15A1 D-Lysine, L-alanyl- 30000000 NA NA NA NA NA TTD
SLC15A1 (2S)-2-amino-5-[[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy]-5-oxopentanoic acid NA 11450000 NA NA NA NA BindingDB
SLC15A1 (2S)-2-amino-4-[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)oxolan-3-yl]oxy-4-oxobutanoic acid NA 13920000 NA NA NA NA BindingDB
SLC15A1 (2S)-2-amino-5-[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)oxolan-3-yl]oxy-5-oxopentanoic acid NA 12980000 NA NA NA NA BindingDB
SLC15A1 (2S)-2-amino-4-[[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy]-4-oxobutanoic acid NA 10230000 NA NA NA NA BindingDB
SLC15A1 [(2R,3S,5R)-3-[(2S)-2-amino-3-methylbutanoyl]oxy-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methyl (2S)-2-amino-3-methylbutanoate NA 2240000 NA NA NA NA BindingDB
SLC15A1 (2S)-3-hydroxy-2-[[(2S,4S)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid NA 9800000 NA NA NA NA BindingDB
SLC15A1 (2R)-3-hydroxy-2-[[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid NA 10200000 NA NA NA NA BindingDB
SLC15A1 (2S)-3-hydroxy-2-[[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid NA 9600000 NA NA NA NA BindingDB
SLC15A1 2-amino-N-(3-phenylphenyl)propanamide 290000 NA NA NA NA NA TTD
SLC15A1 Dicloxacillin 7200000 NA NA NA NA NA BindingDB|PubChem|TTD
SLC15A1 3-[(2-Ammoniopropanoyl)amino]benzoate 310000 NA NA NA NA NA TTD
SLC15A1 Cyclacillin NA|500000 350000|600000|NA NA NA NA NA BindingDB|PubChem|TTD
SLC15A1 Prolylglutamic acid NA|20000000 12300000|NA NA NA|5000000 NA NA BindingDB|TTD
SLC15A1 H-D-Ala-DL-Ala-OH 4200000 NA NA NA NA NA BindingDB