GENE_SYMBOL |
DRUG_NAME |
Ki (nM) |
IC50 (nM) |
Kd (nM) |
EC50 (nM) |
Potency (nM) |
AC50 (nM) |
Datasource |
SLC15A1 |
Arg-Arg |
NA |
7310000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Pro-Tyr |
730000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Ala-Ser |
140000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
Glycyl-L-alanine |
NA |
NA|1820000 |
NA |
520000|NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
[(3S,7R,8aS)-7-hydroxy-1,4-dioxo-2,3,6,7,8,8a-hexahydropyrrolo[1,2-a]pyrazin-3-yl]methyl (2S)-2-amino-3-methylbutanoate |
NA |
2900000 |
NA |
NA |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
D-Lysine, L-alanyl- |
30000000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
(2S)-2-amino-5-[[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy]-5-oxopentanoic acid |
NA |
11450000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2S)-2-amino-4-[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)oxolan-3-yl]oxy-4-oxobutanoic acid |
NA |
13920000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2S)-2-amino-5-[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-2-(hydroxymethyl)oxolan-3-yl]oxy-5-oxopentanoic acid |
NA |
12980000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2S)-2-amino-4-[[(2R,3S,5R)-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)-3-hydroxyoxolan-2-yl]methoxy]-4-oxobutanoic acid |
NA |
10230000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
[(2R,3S,5R)-3-[(2S)-2-amino-3-methylbutanoyl]oxy-5-(5-fluoro-2,4-dioxopyrimidin-1-yl)oxolan-2-yl]methyl (2S)-2-amino-3-methylbutanoate |
NA |
2240000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2S)-3-hydroxy-2-[[(2S,4S)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid |
NA |
9800000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2R)-3-hydroxy-2-[[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid |
NA |
10200000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
(2S)-3-hydroxy-2-[[(2R,4S)-4-hydroxypyrrolidine-2-carbonyl]amino]propanoic acid |
NA |
9600000 |
NA |
NA |
NA |
NA |
BindingDB |
SLC15A1 |
2-amino-N-(3-phenylphenyl)propanamide |
290000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Dicloxacillin |
7200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC15A1 |
3-[(2-Ammoniopropanoyl)amino]benzoate |
310000 |
NA |
NA |
NA |
NA |
NA |
TTD |
SLC15A1 |
Cyclacillin |
NA|500000 |
350000|600000|NA |
NA |
NA |
NA |
NA |
BindingDB|PubChem|TTD |
SLC15A1 |
Prolylglutamic acid |
NA|20000000 |
12300000|NA |
NA |
NA|5000000 |
NA |
NA |
BindingDB|TTD |
SLC15A1 |
H-D-Ala-DL-Ala-OH |
4200000 |
NA |
NA |
NA |
NA |
NA |
BindingDB |