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Drugs And Genes
Negative Drug Target Genes
Gene
Drug
GENE_SYMBOL
DRUG_NAME
Ki (nM)
IC50 (nM)
Kd (nM)
EC50 (nM)
Potency (nM)
AC50 (nM)
Datasource
SLC15A1
2-[[(2S)-2-aminopropanoyl]amino]-2-methylpropanoic acid
1200000
NA
NA
NA
NA
NA
TTD
SLC15A1
(S)-6-Amino-2-((R)-2-amino-propionylamino)-hexanoic acid
7000000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
5-Amino-2-(2-amino-propionylamino)-pentanoic acid
970000
NA
NA
NA
NA
NA
BindingDB
SLC15A1
N-(L-Alanyl)-N-methylglycine
250000
NA
NA
NA
NA
NA
TTD
SLC15A1
Alanyl ornithine
970000
NA
NA
NA
NA
NA
TTD
SLC15A1
Floxacillin
3200000
NA
NA
NA
NA
NA
BindingDB|PubChem|TTD
SLC15A1
4-[(2-Ammoniopropanoyl)amino]benzoate
9100000
NA
NA
NA
NA
NA
TTD
SLC15A1
[3-(Hydroxymethyl)phenyl]guanidine
NA
3000000
NA
NA
NA
NA
TTD
SLC15A1
5'-Val-Floxuridine
NA
1120000
NA
NA
NA
NA
BindingDB
SLC15A1
3-Methyl-1-oxo-1-piperidin-1-ylpentan-2-aminium
5620000
NA
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
2-amino-N-(3-methylphenyl)propanamide
410000
NA
NA
NA
NA
NA
TTD
SLC15A1
2-amino-N-(3-chlorophenyl)propanamide
460000
NA
NA
NA
NA
NA
TTD
SLC15A1
2-amino-N-(2-chlorophenyl)propanamide
7800000
NA
NA
NA
NA
NA
TTD
SLC15A1
(S)-2-((S)-2-amino-3-(2,5,7-tri-tert-butyl-1H-indol-3-yl)propanamido)-5-guanidinopentanamide
NA
600000
NA
NA
NA
NA
BindingDB|TTD
SLC15A1
2-[(2-Ammoniopropanoyl)amino]pentanedioate
320000
NA
NA
NA
NA
NA
BindingDB
SLC15A1
[(2-Ammonio-3-mercaptopropanoyl)amino]acetate
200000
NA
NA
NA
NA
NA
BindingDB
SLC15A1
3-(3-Aminopropanoylamino)propanoic acid
30000000
NA
NA
NA
NA
NA
TTD
SLC15A1
Cephalexin
NA|14000000|14400000
5200000|13700000|NA
NA
NA
NA
NA
BindingDB|PubChem|TTD
SLC15A1
N-biphenyl-2-ylalaninamide
16600000
NA
NA
NA
NA
NA
TTD
SLC15A1
N-glycylproline
NA|300000
NA|330000
NA
130000|NA
NA
NA
BindingDB|PubChem|TTD
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